SCHEMBL7123218

SCHEMBL7123218

COc1ccc(C(C#N)(CCC(=O)O)C(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CYP3A4 P08684 5/20 0.43
PDE4B Q07343 1/20 0.41
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KIF11 P52732 1/20 0.40
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 2/20 0.39
HSD17B10 Q99714 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FFAR1 O14842 1/20 0.39
ABCB1 P08183 5/20 0.39
CYP3A5 P20815 1/20 0.38
EBP Q15125 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5751980 0.84 EBP (0.51) CYP3A4NPSR1KIF11MAPTALDH1A1
SCHEMBL7123137 0.83 EBP (0.40) CYP3A4ALDH1A1FFAR1ABCB1EBP
SCHEMBL7131765 0.83 MMP2 (0.41) CYP3A4HTTKIF11GAAMAPT
SCHEMBL7120088 0.83 EBP (0.40) CYP3A4ALDH1A1HSD17B10ABCB1CYP3A5
SCHEMBL7128373 0.83 MIF (0.41) NPC1RAB9ACYP3A4ALDH1A1L3MBTL1
SCHEMBL7126244 0.83 EBP (0.40) CYP3A4HTTALDH1A1FFAR1ABCB1
SCHEMBL7751300 0.83 CYP3A4 (0.63) CYP3A4HTTNPSR1GAAMAPT
SCHEMBL7132572 0.83 CYP3A4 (0.63) CYP3A4HTTNPSR1GAAMAPT
SCHEMBL11091478 0.80 NPC1 (0.46) NPC1RAB9ACYP3A4PDE4BHTT
SCHEMBL5753427 0.80 CYP3A4 (0.43) NPC1RAB9ACYP3A4HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US claimed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP claimed
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US disclosed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP disclosed