SCHEMBL7126078

SCHEMBL7126078

O=C(NC(Cc1ccc(C(F)(F)F)cc1)C(O)c1ccc2ccccc2c1)c1cccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.48
MCHR1 Q99705 1/20 0.47
UTS2R Q9UKP6 3/20 0.46
PIN1 Q13526 2/20 0.45
RXFP1 Q9HBX9 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
BACE1 P56817 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
PTGER4 P35408 1/20 0.40
PTGDR Q13258 1/20 0.40
CNR2 P34972 1/20 0.39
P2RX1 P51575 1/20 0.39
P2RX3 P56373 1/20 0.39
P2RX4 Q99571 1/20 0.39
P2RX7 Q99572 1/20 0.39
CCR3 P51677 1/20 0.39
HDAC8 Q9BY41 2/20 0.39
MMP3 P08254 1/20 0.39
HDAC3 O15379 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752263 0.89 DRD4 (0.48) DRD4MCHR1PIN1RXFP1ALDH1A1
SCHEMBL5751220 0.89 DRD4 (0.48) DRD4MCHR1PIN1RXFP1ALDH1A1
SCHEMBL5751363 0.86 DRD4 (0.51) DRD4MCHR1PIN1RXFP1ALDH1A1
SCHEMBL5750142 0.85 DRD4 (0.40) DRD4MCHR1UTS2RPIN1BACE1
SCHEMBL5753845 0.83 DRD4 (0.41) DRD4MCHR1TRPV1PTGER4PTGDR
SCHEMBL5753159 0.82 DRD4 (0.39) DRD4MCHR1UTS2RPIN1PTGER4
SCHEMBL5752112 0.82 DRD4 (0.50) DRD4MCHR1PIN1RXFP1BACE1
SCHEMBL5752865 0.81 PIN1 (0.57) DRD4MCHR1PIN1HDAC8HDAC3
SCHEMBL5753785 0.81 HDAC8 (0.46) ALDH1A1LMNABACE1CNR2CCR3
SCHEMBL5754521 0.80 MCHR1 (0.48) DRD4MCHR1BACE1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed