SCHEMBL7127720

SCHEMBL7127720

COC(=O)/C=C(/C)N1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
ALOX12 P18054 1/20 0.44
MAPT P10636 1/20 0.41
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
HPGD P15428 2/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5996600 1.00 ALDH1A1 (0.44) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL7877240 1.00 ALDH1A1 (0.44) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL535867 0.79 NPSR1 (0.46) ALDH1A1USP2LMNAALOX12HCAR2
SCHEMBL106944 0.79 NPSR1 (0.46) ALDH1A1USP2LMNAALOX12HCAR2
SCHEMBL1778153 0.79 NPSR1 (0.46) ALDH1A1USP2LMNAALOX12HCAR2
SCHEMBL10583065 0.78 ALDH1A1 (0.49) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL22783869 0.78 ALDH1A1 (0.49) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL10583061 0.78 ALDH1A1 (0.49) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL7975644 0.77 NPSR1 (0.44) ALDH1A1USP2LMNAALOX12MAPT
SCHEMBL11719535 0.77 NPSR1 (0.44) ALDH1A1USP2LMNAALOX12MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6586613-B1 Compounds such as 5-(tert-butyldimethylsiloxy)-7,7-dimethyl -4(4-fluorophenyl)-3-(hydroxy-(4-trifluorophenyl)-methyl)-2-isopropyl -5,6,7,8-tetrahydronaphthalene, used as antagonists for cholesteryl ester transferase protein; hyperlipemia BAYER AKTIENGELLSCHAFT (DE) 2003-07-01 US disclosed