SCHEMBL7133997

SCHEMBL7133997

O=C1Nc2c(Br)cc(Br)cc2C1=Cc1cccc(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
FLT3 P36888 2/20 0.38
MAP1LC3B Q9GZQ8 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
XBP1 P17861 1/20 0.35
MAPK1 P28482 1/20 0.35
NTSR1 P30989 1/20 0.35
RPS6KA3 P51812 1/20 0.35
RET P07949 1/20 0.34
PDGFRB P09619 1/20 0.34
CDK2 P24941 1/20 0.34
KDR P35968 1/20 0.34
PLK4 O00444 1/20 0.34
PLK1 P53350 1/20 0.34
SIRT1 Q96EB6 2/20 0.34
RAF1 P04049 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7139764 0.90 NPC1 (0.57) NPC1KMT2AMEN1FLT3MAP1LC3B
SCHEMBL7134446 0.88 NPC1 (0.43) NPC1KMT2AMEN1FLT3MAP1LC3B
SCHEMBL5362288 0.86 CES1 (0.39) NPC1KMT2AMEN1FLT3MAP1LC3B
SCHEMBL5365774 0.83 IKBKB (0.41) NPC1KMT2AMEN1ALDH1A1MAPT
SCHEMBL7136542 0.81 FLT3 (0.43) NPC1KMT2AMEN1FLT3MAP1LC3B
SCHEMBL7136300 0.80 MAP3K7 (0.45) KMT2AMEN1MAP1LC3BALDH1A1MAPT
SCHEMBL7134869 0.80 SIRT1 (0.43) NPC1KMT2AMEN1ALDH1A1MAPT
SCHEMBL7139735 0.80 KMT2A (0.55) NPC1KMT2AMEN1FLT3ALDH1A1
SCHEMBL5362880 0.80 PLK4 (0.57) KMT2AMEN1FLT3MAP1LC3BALDH1A1
SCHEMBL7140941 0.79 MYC (0.43) NPC1KMT2AMEN1FLT3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed