SCHEMBL7138178

SCHEMBL7138178

Cc1c(Br)cc(Br)c2c1C(=Cc1c(F)cccc1C(F)(F)F)C(=O)N2

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
XBP1 P17861 1/20 0.34
MAPK1 P28482 1/20 0.34
NTSR1 P30989 1/20 0.34
KMT2A Q03164 1/20 0.34
MAP4K1 Q92918 4/20 0.33
HTR2C P28335 4/20 0.31
HTR2B P41595 4/20 0.31
HTR2A P28223 3/20 0.31
FLT3 P36888 1/20 0.31
STK10 O94804 1/20 0.30
SLK Q9H2G2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7131380 0.90 IKBKB (0.35) ALDH1A1MAPTXBP1MAPK1NTSR1
SCHEMBL7134217 0.85 CES1 (0.35) CES1ALDH1A1MAPTXBP1MAPK1
SCHEMBL5366373 0.83 KDR (0.36) KMT2AHTR2CHTR2BHTR2AFLT3
SCHEMBL7140036 0.83 MYC (0.42) CES1ALDH1A1MAPTXBP1MAPK1
SCHEMBL5358358 0.80 CES1 (0.39) CES1ALDH1A1MAPTXBP1MAPK1
SCHEMBL7135758 0.80 NPC1 (0.38) ALDH1A1MAPTXBP1MAPK1NTSR1
SCHEMBL7138946 0.79 NPC1 (0.48) ALDH1A1MAPTXBP1MAPK1NTSR1
SCHEMBL7136928 0.79 KMT2A (0.37) ALDH1A1MAPTXBP1MAPK1NTSR1
SCHEMBL7133731 0.79 PTP4A3 (0.38) ALDH1A1MAPTXBP1MAPK1NTSR1
SCHEMBL7131271 0.78 ERN1 (0.38) ALDH1A1MAPTXBP1MAPK1NTSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed