SCHEMBL7140036

SCHEMBL7140036

Cc1c(Br)cc(Br)c2c1C(=Cc1ccccc1C(F)(F)F)C(=O)N2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.42
MAX P61244 1/20 0.42
TNF P01375 3/20 0.38
IL6 P05231 2/20 0.38
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
XBP1 P17861 1/20 0.36
MAPK1 P28482 1/20 0.36
NTSR1 P30989 1/20 0.36
MEN1 O00255 2/20 0.36
CES1 P23141 1/20 0.35
CYP24A1 Q07973 1/20 0.34
RAB9A P51151 1/20 0.33
NOD1 Q9Y239 1/20 0.33
PTPN1 P18031 1/20 0.33
NFKB1 P19838 1/20 0.33
ADORA2A P29274 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7134217 0.90 CES1 (0.35) MYCMAXKDM4EKMT2AALDH1A1
SCHEMBL7136928 0.86 KMT2A (0.37) KMT2AALDH1A1MAPTXBP1MAPK1
SCHEMBL7138169 0.85 POLB (0.42) KMT2AALDH1A1MAPTXBP1MAPK1
SCHEMBL7138946 0.84 NPC1 (0.48) KDM4EKMT2AALDH1A1MAPTXBP1
SCHEMBL7139425 0.84 KMT2A (0.49) KDM4EKMT2AALDH1A1MAPTXBP1
SCHEMBL7138178 0.83 CES1 (0.35) KMT2AALDH1A1MAPTXBP1MAPK1
SCHEMBL7134441 0.82 MYC (0.43) MYCMAXTNFIL6KMT2A
SCHEMBL7134889 0.82 DYRK1A (0.39) KMT2AALDH1A1MAPTXBP1MAPK1
SCHEMBL7134752 0.82 PLK4 (0.48) KMT2AALDH1A1MAPTXBP1MAPK1
SCHEMBL7135758 0.80 NPC1 (0.38) KDM4EKMT2AALDH1A1MAPTXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed