SCHEMBL7138236

SCHEMBL7138236

Cc1c(Br)cc(Br)c2c1C(=Cc1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1)C(=O)N2

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.51
ERBB2 P04626 1/20 0.51
IGF1R P08069 1/20 0.51
EEF2K O00418 1/20 0.49
SRC P12931 1/20 0.49
GAA P10253 2/20 0.48
CTRC Q99895 1/20 0.47
PTGS2 P35354 7/20 0.46
PTGS1 P23219 4/20 0.46
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7137523 0.95 ERBB2 (0.46) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7138387 0.94 EGFR (0.46) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7133835 0.92 ERBB2 (0.44) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7137037 0.89 KMT2A (0.42) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7135662 0.87 ERBB2 (0.41) EGFRERBB2IGF1RCTRCPTGS2
SCHEMBL7139429 0.86 ERBB2 (0.53) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7133862 0.85 EEF2K (0.47) EGFREEF2KSRCGAACYP1A2
SCHEMBL7134037 0.85 MAP1LC3B (0.45) EGFRCYP1A2CYP2C9MEN1KMT2A
SCHEMBL7136796 0.84 TDP1 (0.37) EGFRERBB2IGF1REEF2KSRC
SCHEMBL7132027 0.84 ERBB2 (0.60) EGFRERBB2IGF1REEF2KSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506763-B2 Useful in prevention and treatment of protein kinase related disorders such as cancer SUGEN, INC. 2003-01-14 US disclosed