SCHEMBL7140048

SCHEMBL7140048

CCc1nn2c(N)cc(C)nc2c1S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 14/20 0.58
ALDH1A1 P00352 2/20 0.45
PKM P14618 2/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
POLB P06746 1/20 0.43
RAPGEF4 Q8WZA2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136436 0.87 HTR6 (0.58) HTR6ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL7136288 0.85 HTR6 (0.80) HTR6
SCHEMBL7133537 0.81 HTR6 (0.57) HTR6ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL7141435 0.80 HTR6 (0.51) HTR6ALDH1A1HPGDSMN1; SMN2CYP3A4
SCHEMBL7133638 0.80 HTR6 (0.50) HTR6ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL7133635 0.80 HTR6 (0.50) HTR6ALDH1A1KDM4EHPGDCYP3A4
SCHEMBL7134457 0.74 HTR6 (0.52) HTR6
SCHEMBL13016796 0.73 HTR6 (1.00) HTR6
SCHEMBL7134508 0.73 HTR6 (0.48) HTR6
SCHEMBL13016798 0.73 HTR6 (1.00) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941994-B1 Pyrazolopyrimidines and pyrazolotriazines with 5-HT6 receptor affinity HOFFMANN LA ROCHE (CH) 2003-05-14 EP disclosed
US-6194410-B1 ANTISEROTONINE AGENTS; NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS HOFFMAN-LA ROCHE INC. 2001-02-27 US disclosed
EP-0941994-A1 Pyrazolopyrimidines and pyrazolotriazines with 5-HT6 receptor affinity F. HOFFMANN-LA ROCHE AG (CH) 1999-09-15 EP disclosed