SCHEMBL7140885

SCHEMBL7140885

Cc1cccc(C2c3ccccc3C=NN2C=CC=O)n1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 7/20 0.35
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144192 0.81 HHAT (0.33) HHATALDH1A1HPGDMEN1KMT2A
SCHEMBL7136528 0.80 DRD2 (0.33)
SCHEMBL7140432 0.79 HHAT (0.36) HHATALDH1A1MEN1KMT2A
SCHEMBL7136773 0.78
SCHEMBL7142692 0.78
SCHEMBL7143190 0.78
SCHEMBL7142153 0.78
SCHEMBL7137225 0.76 MAPT (0.32)
SCHEMBL7138487 0.76 MAPT (0.32)
SCHEMBL7143865 0.76 MAPT (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966464-B1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-05-28 EP disclosed
US-6114330-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 2000-09-05 US disclosed
EP-0966464-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1999-12-29 EP disclosed
WO-1998039328-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F.HOFFMANN-LA ROCHE AG (CH) 1998-09-11 WO disclosed