SCHEMBL7141306

SCHEMBL7141306

CSc1nn2c(Cl)c(C)c(C)nc2c1S(=O)(=O)c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 20/20 0.75
HTR2B P41595 2/20 0.63
KCNH2 Q12809 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12426989 0.86 HTR6 (1.00) HTR6HTR2BKCNH2
SCHEMBL12427475 0.81 HTR6 (1.00) HTR6HTR2BKCNH2
SCHEMBL12428302 0.81 HTR6 (0.75) HTR6HTR2BKCNH2
SCHEMBL7136536 0.81 HTR6 (0.78) HTR6HTR2BKCNH2
SCHEMBL7135365 0.80 HTR6 (0.67) HTR6HTR2BKCNH2
SCHEMBL7136576 0.80 HTR6 (0.60) HTR6HTR2BKCNH2
SCHEMBL7139046 0.80 HTR6 (0.66) HTR6HTR2BKCNH2
SCHEMBL7136399 0.79 HTR6 (0.60) HTR6HTR2BKCNH2
SCHEMBL12427333 0.79 HTR6 (0.72) HTR6HTR2BKCNH2
SCHEMBL7140510 0.79 HTR6 (0.79) HTR6HTR2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941994-B1 Pyrazolopyrimidines and pyrazolotriazines with 5-HT6 receptor affinity HOFFMANN LA ROCHE (CH) 2003-05-14 EP disclosed
US-6194410-B1 ANTISEROTONINE AGENTS; NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS HOFFMAN-LA ROCHE INC. 2001-02-27 US disclosed
EP-0941994-A1 Pyrazolopyrimidines and pyrazolotriazines with 5-HT6 receptor affinity F. HOFFMANN-LA ROCHE AG (CH) 1999-09-15 EP disclosed