SCHEMBL7141490

SCHEMBL7141490

Fc1ccc([C@H]2NN=Cc3ccccc32)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.38
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 1/20 0.35
HTR1A P08908 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
IDO1 P14902 2/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
MC4R P32245 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141484 1.00 JAK2 (0.38) JAK2KDM4EPOLBMAPTALOX15
SCHEMBL7142187 0.80 PRCP (0.44) JAK2MAPTHTR2AHTR2CHTR2B
SCHEMBL7142182 0.80 PRCP (0.44) JAK2MAPTHTR2AHTR2CHTR2B
SCHEMBL4273310 0.72 HTR2C (0.41) HTR2AHTR2CHTR2B
SCHEMBL7138440 0.72 PRCP (0.38) KDM4EMAPTHSD17B10
SCHEMBL7142141 0.70 HTR2C (0.41) KDM4EALOX15HSD17B10HTR2AHTR2C
SCHEMBL7142143 0.70 HTR2C (0.41) KDM4EALOX15HSD17B10HTR2AHTR2C
SCHEMBL7135564 0.69 PRCP (0.33)
SCHEMBL7135566 0.69 PRCP (0.33)
SCHEMBL4273307 0.68 PRCP (0.45) KDM4EMAPTALOX15HSD17B10SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966464-B1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-05-28 EP disclosed
US-6114330-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 2000-09-05 US disclosed
EP-0966464-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1999-12-29 EP disclosed
WO-1998039328-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F.HOFFMANN-LA ROCHE AG (CH) 1998-09-11 WO disclosed