SCHEMBL7142143

SCHEMBL7142143

Cc1cccc([C@@H]2NN=Cc3ccccc32)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.41
MAOB P27338 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HDAC4 P56524 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
HTR2B P41595 1/20 0.35
SLC6A3 Q01959 1/20 0.35
NPC1 O15118 1/20 0.35
HPN P05981 1/20 0.35
HSD17B10 Q99714 1/20 0.34
PKM P14618 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP19A1 P11511 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142141 1.00 HTR2C (0.41) HTR2CMAOBKDM4EMEN1KMT2A
SCHEMBL7135564 0.88 PRCP (0.33)
SCHEMBL7135566 0.88 PRCP (0.33)
SCHEMBL4273307 0.84 PRCP (0.45) MAOBKDM4EMEN1KMT2AHDAC4
SCHEMBL7138440 0.82 PRCP (0.38) KDM4EMEN1KMT2AALDH1A1GAA
SCHEMBL7142700 0.82 DRD2 (0.33) HTR2CALDH1A1HTR2AHTR2BDRD2
SCHEMBL7139594 0.77 CYP1A2 (0.33) HTR2C
SCHEMBL4273310 0.76 HTR2C (0.41) HTR2CMAOBALDH1A1HTR2AHTR2B
SCHEMBL7138973 0.75 HSP90AA1 (0.43) KDM4EALDH1A1GAANPC1
SCHEMBL7138978 0.75 HSP90AA1 (0.43) KDM4EALDH1A1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966464-B1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES BASILEA PHARMACEUTICA AG (CH) 2003-05-28 EP disclosed
US-6114330-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 2000-09-05 US disclosed
EP-0966464-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1999-12-29 EP disclosed
WO-1998039328-A1 SUBSTITUTED 2,4-DIAMINOPYRIMIDINES F.HOFFMANN-LA ROCHE AG (CH) 1998-09-11 WO disclosed