SCHEMBL7141540

SCHEMBL7141540

CON=C(C(=O)OC)c1ccccc1C=CC=Cc1ccccc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.53
NFKB1 P19838 1/20 0.46
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 2/20 0.44
GAA P10253 1/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NFE2L2 Q16236 1/20 0.41
MAOA P21397 1/20 0.40
BACE1 P56817 1/20 0.40
P4HB P07237 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141534 1.00 MAOB (0.53) MAOBNFKB1LMNAMAPTMEN1
SCHEMBL7141537 1.00 MAOB (0.53) MAOBNFKB1LMNAMAPTMEN1
SCHEMBL9238440 0.83 HIF1A (0.44) MAOBHIF1ANFE2L2BACE1
SCHEMBL9236683 0.82 HIF1A (0.45) MAOBHIF1ANFE2L2BACE1
SCHEMBL9239702 0.78 KDM4E (0.50) MAOBLMNAMAPTKMT2AHIF1A
SCHEMBL8954615 0.78 HIF1A (0.47) LMNAHIF1ANFE2L2BACE1
SCHEMBL8835428 0.77 HIF1A (0.48) LMNAMAPTMEN1KMT2AHIF1A
SCHEMBL7206001 0.77 HIF1A (0.48) LMNAMAPTMEN1KMT2AHIF1A
SCHEMBL7209021 0.77 HIF1A (0.48) LMNAMAPTMEN1KMT2AHIF1A
SCHEMBL9239168 0.76 HIF1A (0.43) MAOBLMNAHIF1ANFE2L2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP disclosed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US disclosed