SCHEMBL7142022

SCHEMBL7142022

CO/C=C(/C(=O)O)c1ccccc1/C=C/C=C/c1ccc2ccccc2c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.42
CAPN1 P07384 2/20 0.42
CNR2 P34972 2/20 0.41
MAOB P27338 1/20 0.41
NQO2 P16083 2/20 0.41
RELA Q04206 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
APP P05067 1/20 0.40
MAPT P10636 1/20 0.40
PTGS1 P23219 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7142025 1.00 AKR1C3 (0.42) AKR1C3CAPN1CNR2MAOBNQO2
SCHEMBL7142028 1.00 AKR1C3 (0.42) AKR1C3CAPN1CNR2MAOBNQO2
SCHEMBL7139094 0.86 MAOB (0.42) MAOB
SCHEMBL7139096 0.86 MAOB (0.42) MAOB
SCHEMBL7143682 0.85 MAOB (0.52) MAOBRELAMAPT
SCHEMBL7143686 0.85 MAOB (0.52) MAOBRELAMAPT
SCHEMBL7140078 0.83 TUBB4A (0.40) MAOB
SCHEMBL7136432 0.83 MAOB (0.46) MAOBMAPT
SCHEMBL7140080 0.83 TUBB4A (0.40) MAOB
SCHEMBL7136433 0.83 MAOB (0.46) MAOBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996439-B1 BETA-ALKOXYACRYLATES AGAINST MALARIA HOFFMANN LA ROCHE (CH) 2003-01-08 EP disclosed
US-6084120-A ACTIVE AGAINST CHLOROQUINE-SENSITIVE PATIENTS AND AGAINST CHLOROQUINE-RESISTANT MALARIA PATHOGENS; PROPHYLAXIS AND TREATMENT; E.G., A 3 METHOXY-2-(2-(4-PHENYLBUTA-1,3-DIEN-1-YL)PHENYL)ACRYLIC ACID HOFFMANN-LA ROCHE INC. (US) 2000-07-04 US disclosed