Benzoic Acid

Benzoic Acid

SCHEMBL7142175

Cc1[nH]c2ccc(N(C(N)=S)c3cccc(-c4ccccc4)c3)cc2c1CCN(C)Cc1cc(N(C)C)cnn1.O=C(O)c1ccccc1

nearest known ligand 0.34

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CACNA1CCACNA1DCACNA1FCACNA1SDPP4HTR1BHTR1D

The experimentally established mechanism targets of Benzoic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.34
ALDH1A1 P00352 4/20 0.34
MAPK1 P28482 1/20 0.34
HTR1F P30939 1/20 0.33
NPSR1 Q6W5P4 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 7/20 0.32
MEN1 O00255 6/20 0.32
ATM Q13315 4/20 0.32
GAA P10253 3/20 0.32
KDM4E B2RXH2 2/20 0.32
PPARG P37231 1/20 0.32
PSMD14 O00487 1/20 0.32
RECQL P46063 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
RAB9A P51151 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoic Acid SCHEMBL7141730 0.94 HTR1F (0.34) MAPTALDH1A1MAPK1HTR1FNPSR1
Benzoic Acid SCHEMBL8552961 0.86 MEN1 (0.30) MAPK1KMT2AMEN1
Benzoic Acid SCHEMBL8548262 0.86
Benzoic Acid SCHEMBL8549809 0.81 FYN (0.31)
Benzoic Acid SCHEMBL8551806 0.81 MEN1 (0.31) MAPK1NPSR1KMT2AMEN1LMNA
Benzoic Acid SCHEMBL8191205 0.78 HTR1F (0.45) MAPTALDH1A1MAPK1HTR1FNPSR1
Benzoic Acid SCHEMBL7141174 0.75 HTR1F (0.41) MAPTALDH1A1HTR1FSMN1; SMN2KMT2A
Benzoic Acid SCHEMBL8436196 0.72 PDPK1 (0.33) MAPK1
Benzoic Acid SCHEMBL8435537 0.70 PDPK1 (0.33) MAPTMAPK1LMNA
Benzoic Acid SCHEMBL8709658 0.69 TMEM97 (0.33) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0768301-B1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists LILLY CO ELI (US) 2003-04-02 EP disclosed
US-6126932-A INSOLUBLE POLYMER BEARING PENDANT SIDE CHAINS, SAID SIDE CHAINS EACH TERMINATING WITH THE 1-(3-(1-PYRROLIDINYL)-PROPYL)-3-ETHYLCARBODIIMIDE MOIETY. ELI LILLY AND COMPANY (US) 2000-10-03 US disclosed
EP-0994109-A2 1-(3-(1-Pyrrolidinyl)propyl)-3-ethylcarbodiimide and a solid phase coupling agent ELI LILLY AND COMPANY (US) 2000-04-19 EP disclosed
US-5998630-A A 1-(3-(1-PYRROLIDINYL)PROPY)-3-ETHYLCARBODIIMIDE ELI LILLY AND COMPANY (US) 1999-12-07 US disclosed
EP-0768301-A1 N-(2-substituted-3-(2-aminoethyl)-1H-indol-5-yl)-amides as new 5-HT1F agonists ELI LILLY AND COMPANY (US) 1997-04-16 EP disclosed