SCHEMBL7142800

SCHEMBL7142800

C=CC(=O)N(c1ccccc1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
TRPM8 Q7Z2W7 2/20 0.37
TGM2 P21980 1/20 0.36
CES1 P23141 2/20 0.35
ALDH1A1 P00352 4/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
TSHR P16473 2/20 0.33
MEN1 O00255 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR1H3 Q13133 1/20 0.33
MLYCD O95822 1/20 0.33
POLQ O75417 1/20 0.33
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7891310 0.81 CYP2C19 (0.41) AKT1NPSR1TRPM8TGM2ALDH1A1
SCHEMBL3938034 0.80 NPSR1 (0.43) NPSR1CES1ALDH1A1CYP3A4CYP2C9
SCHEMBL27490821 0.80 ALDH1A1 (0.40) AKT1NPSR1TRPM8TGM2ALDH1A1
SCHEMBL1008397 0.78 NPSR1 (0.44) NPSR1CES1ALDH1A1CYP3A4CYP2C9
SCHEMBL21392794 0.76 KMT2A (0.40) AKT1ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL6611167 0.75 AKT1 (0.43) AKT1NPSR1TRPM8TGM2ALDH1A1
SCHEMBL1067570 0.75 NPSR1 (0.41) NPSR1CES1ALDH1A1CYP3A4CYP2C9
SCHEMBL7827701 0.75 NPSR1 (0.41) NPSR1TRPM8CES1ALDH1A1CYP3A4
SCHEMBL28247945 0.75 NPSR1 (0.41) NPSR1CES1ALDH1A1CYP3A4CYP2C9
SCHEMBL11370851 0.75 NPSR1 (0.41) NPSR1CES1ALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730454-A4 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO INC (US) 2003-06-04 EP disclosed
EP-0730454-A1 ANTIARRHYTHMIC BENZODIAZEPINES MERCK & CO. INC. (US) 1996-09-11 EP disclosed