SCHEMBL7144539

SCHEMBL7144539

COc1c(C(N)=O)cc(-c2cccc(NC(C)=O)c2)n2n[c]nc12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FYN P06241 15/20 0.46
BRAF P15056 2/20 0.42
PI4K2A Q9BTU6 1/20 0.41
PARP1 P09874 1/20 0.41
DHODH Q02127 1/20 0.41
PAX8 Q06710 1/20 0.40
DYRK3 O43781 1/20 0.40
CCNT1 O60563 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CDK9 P50750 1/20 0.40
CDK5 Q00535 1/20 0.40
DYRK1A Q13627 1/20 0.40
CDK5R1 Q15078 1/20 0.40
DYRK2 Q92630 1/20 0.40
DYRK1B Q9Y463 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146854 0.87 PDE4D (0.43) FYN
SCHEMBL7043840 0.85 PARP1 (0.43) FYNPARP1
SCHEMBL7146568 0.85 IKBKB (0.38) FYNPARP1
SCHEMBL14888540 0.85 FYN (0.46) FYNPI4K2APARP1DHODHDYRK3
SCHEMBL7145673 0.85 TLR8 (0.48) FYNPARP1DHODH
SCHEMBL7041861 0.84 IKBKB (0.46) DYRK1B
SCHEMBL6876511 0.84 FYN (0.37) FYN
SCHEMBL7150015 0.81 KDM4E (0.49) FYNBRAFPARP1DYRK3CCNT1
SCHEMBL7041042 0.80 HPGD (0.39) FYN
SCHEMBL7144535 0.79 NTRK1 (0.40) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514989-B1 Has a good affinity to the adenosine receptor and can therefore be used for the treatment or protection of diseases mediated by this receptor HOFFMANN-LA ROCHE INC. 2003-02-04 US disclosed