SCHEMBL7145277

SCHEMBL7145277

CCN1CCN(CCl)C(=O)C1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.34
ALOX15 P16050 1/20 0.33
HTT P42858 1/20 0.32
F2 P00734 1/20 0.31
ELANE P08246 1/20 0.31
CTSG P08311 1/20 0.31
CTRC Q99895 1/20 0.31
INMT O95050 1/20 0.31
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12566554 0.87 GAA (0.48) GAAL3MBTL1POLBSMN1; SMN2ALOX15
Methylene Chloride SCHEMBL29003610 0.80 GAA (0.39) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL28533846 0.79 GAA (0.41) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL12545892 0.77 PIK3CD (0.48) GAAL3MBTL1POLBSMN1; SMN2P2RX7
SCHEMBL7148826 0.76 GAA (0.46) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL10967106 0.76 GAA (0.42) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL12208453 0.76 GAA (0.42) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL7139392 0.76 GAA (0.42) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL12709502 0.76 GAA (0.42) GAAL3MBTL1POLBSMN1; SMN2ALOX15
SCHEMBL22017935 0.76 GAA (0.39) GAAL3MBTL1POLBSMN1; SMN2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100800-B1 NOVEL C-2 S/O- AND S/N FORMALDEHYDE ACETAL DERIVATIVES OF CARBAPENEM-3-CARBOXYLIC ACIDS AND THEIR USE AS ANTIBIOTICS AND BETA-LACTAMASE INHIBITORS PFAENDLER HANS RUDOLF PROF (DE) 2003-06-25 EP disclosed
US-6482818-B2 ANTIBIOTIC PFAENDLER HANS RUDOLF (DE) 2002-11-19 US disclosed
US-20010031749-A1 Novel C-2 S/O-and S/N formaldehyde Acetal Derivatives of Carbapenem-3-carboxylic acids and their use as antibiotics and beta-lactamase inhibitors PFAENDLER HANS RUDOLF (DE) 2001-10-18 US disclosed
EP-1100800-A1 NOVEL C-2 S/O- AND S/N FORMALDEHYDE ACETAL DERIVATIVES OF CARBAPENEM-3-CARBOXYLIC ACIDS AND THEIR USE AS ANTIBIOTICS AND BETA-LACTAMASE INHIBITORS Pfaendler, Hans Rudolf, Prof. (DE) 2001-05-23 EP disclosed
WO-2000006574-A1 NOVEL C-2 S/O- AND S/N FORMALDEHYDE ACETAL DERIVATIVES OF CARBAPENEM-3-CARBOXYLIC ACIDS AND THEIR USE AS ANTIBIOTICS AND β-LACTAMASE INHIBITORS PFAENDLER HANS RUDOLF (DE) 2000-02-10 WO disclosed
EP-0976752-A1 C-2 S/O- and S/N-Formaldehyde acetal derivatives of carbapenem antibiotics Pfaendler, Hans Rudolf, Prof. (DE) 2000-02-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010031749-A1 Novel C-2 S/O-and S/N formaldehyde Acetal Derivatives of Carbapenem-3-carboxylic acids and their use as antibiotics and beta-lactamase inhibitors H1-2, SULT1E1, H1-0 GAA 456/4885L3MBTL1 1727/4885POLB 2130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.