SCHEMBL7148326

SCHEMBL7148326

Clc1ccc(-c2ccc(NCCc3ncccn3)cc2-n2ccnc2)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
IDO1 P14902 3/20 0.41
PDE5A O76074 2/20 0.38
CNR1 P21554 2/20 0.37
CNR2 P34972 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CD38 P28907 2/20 0.36
USP2 O75604 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
NOS1 P29475 2/20 0.35
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
FBP1 P09467 1/20 0.35
NOTUM Q6P988 1/20 0.35
ADRA2C P18825 1/20 0.34
CGAS Q8N884 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7148319 0.80 GSK3B (0.50) CDK1GSK3AGSK3BIDO1PDE5A
SCHEMBL6069053 0.70 GSK3B (0.47) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL5089665 0.68 CDK1 (0.51) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL6334824 0.67 IDO1 (0.65) IDO1CNR1CNR2MEN1KMT2A
SCHEMBL29367195 0.67 IDO1 (0.50) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL5089661 0.67 GSK3B (0.60) CDK1GSK3AGSK3BIDO1PDE5A
SCHEMBL5099510 0.65 CNR1 (0.51) CDK1GSK3AGSK3BIDO1PDE5A
SCHEMBL27253612 0.65 CDK1 (0.49) CDK1GSK3AGSK3BIDO1CNR1
SCHEMBL6342180 0.65 IDO1 (0.70) IDO1MEN1KMT2AMAPK1NOTUM
SCHEMBL27538053 0.65 GSK3B (0.56) CDK1GSK3AGSK3BIDO1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed