SCHEMBL7148685

SCHEMBL7148685

Cc1cc(C)cc(C[SiH2]CCOCn2c(C=O)nc3cc(Cl)ccc32)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VDR P11473 2/20 0.39
KMT2A Q03164 2/20 0.36
TBXA2R P21731 5/20 0.34
ALDH1A1 P00352 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTT P42858 1/20 0.34
KCNH2 Q12809 2/20 0.33
KDM4E B2RXH2 2/20 0.32
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
MAPT P10636 1/20 0.31
NUDT1 P36639 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4073539 0.78 VDR (0.45) VDRKMT2ATBXA2RALDH1A1TDP1
SCHEMBL7148680 0.74 VDR (0.42) VDRKMT2ATBXA2RALDH1A1TDP1
SCHEMBL19857776 0.70 NPC1 (0.38) VDRALDH1A1KDM4EP2RX3P2RX2
SCHEMBL19863781 0.68 TBXA2R (0.57) VDRKMT2ATBXA2RALDH1A1TDP1
SCHEMBL3988861 0.64 KDM4E (0.48) VDRKMT2AALDH1A1TDP1KDM4E
SCHEMBL18437170 0.64
SCHEMBL22659127 0.62 KMT2A (0.44) KMT2ATBXA2RALDH1A1TDP1HTT
SCHEMBL31174248 0.61 VDR (0.48) VDRKMT2AALDH1A1TDP1HTT
SCHEMBL31174250 0.61 VDR (0.48) VDRKMT2AALDH1A1TDP1HTT
SCHEMBL900164 0.61 VDR (0.48) VDRKMT2AALDH1A1TDP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317445-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2003-06-11 EP disclosed
WO-2002022600-A2 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2002-03-21 WO disclosed