SCHEMBL7150247

SCHEMBL7150247

COC[C@H]1CCCN1C(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.67
ADORA1 P30542 2/20 0.49
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CAMK1D Q8IU85 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869912 1.00 ADORA2A (0.67) ADORA2AADORA1NPC1RAB9AMEN1
SCHEMBL7150238 1.00 ADORA2A (0.67) ADORA2AADORA1NPC1RAB9AMEN1
SCHEMBL6863273 0.86 ADORA2A (0.71) ADORA2AMEN1KMT2A
SCHEMBL6863643 0.84 ADORA2A (0.73) ADORA2AMEN1KMT2A
SCHEMBL7150287 0.83 ADORA2A (0.65) ADORA2AADORA1NPC1RAB9AMEN1
SCHEMBL6867465 0.83 ADORA2A (0.65) ADORA2AADORA1NPC1RAB9AMEN1
SCHEMBL7150291 0.83 ADORA2A (0.65) ADORA2AADORA1NPC1RAB9AMEN1
SCHEMBL6873056 0.82 ADORA2A (0.65) ADORA2A
SCHEMBL6871917 0.80 ADORA2A (1.00) ADORA2A
SCHEMBL6868028 0.80 ADORA2A (1.00) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US claimed
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed