SCHEMBL7157408

SCHEMBL7157408

Cc1c(C#N)cccc1-c1ccc2c(c1)C(C)(C)OC(=O)N2

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PGR P06401 20/20 0.64
AR P10275 4/20 0.57
NR3C1 P04150 3/20 0.56
NR3C2 P08235 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4175084 0.87 PGR (0.68) PGRARNR3C1NR3C2
SCHEMBL3872645 0.78 PGR (1.00) PGRARNR3C1NR3C2
SCHEMBL4166179 0.78 PGR (0.65) PGRARNR3C1NR3C2
SCHEMBL3876137 0.77 PGR (1.00) PGRARNR3C1NR3C2
SCHEMBL4179192 0.77 PGR (0.82) PGRARNR3C1NR3C2
SCHEMBL3876807 0.76 PGR (0.65) PGRARNR3C1NR3C2
SCHEMBL3870511 0.76 PGR (0.73) PGRARNR3C1NR3C2
SCHEMBL4171050 0.75 PGR (0.69) PGRARNR3C1NR3C2
SCHEMBL3869904 0.75 PGR (1.00) PGRARNR3C1NR3C2
SCHEMBL3883683 0.75 PGR (0.86) PGRARNR3C1NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6509334-B1 This invention relates to compounds that antagonists of the progesterone receptor, their preparation and utility. Intracellular receptors (IR) form a class of structurally related gene regulators known as \"ligand dependent AMERICAN HOME PRODUCTS CORPORATION 2003-01-21 US disclosed