SCHEMBL7157495

SCHEMBL7157495

O=C(O)c1c(C[N+]2(C3CCNCC3)CCCCC2)c(-c2ccccc2)nc2c(F)cccc12

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 12/20 0.43
KCNH2 Q12809 3/20 0.43
GAA P10253 1/20 0.37
TACR2 P21452 2/20 0.37
OPRM1 P35372 1/20 0.37
DHODH Q02127 3/20 0.35
PDE10A Q9Y233 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C8 P10632 1/20 0.34
CYP2C9 P11712 1/20 0.34
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
AURKA O14965 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951612 0.87 TACR3 (0.47) TACR3KCNH2TACR2OPRM1DHODH
Hydrochloric Acid SCHEMBL7077944 0.86 TACR3 (0.47) TACR3KCNH2TACR2OPRM1DHODH
SCHEMBL6582324 0.84 DHODH (0.42) TACR3KCNH2TACR2OPRM1DHODH
Bromide SCHEMBL6953647 0.84 TACR3 (0.34) TACR3KCNH2GAATACR2OPRM1
SCHEMBL6627076 0.84 TACR3 (0.38) TACR3KCNH2TACR2OPRM1DHODH
SCHEMBL7159967 0.83 DHODH (0.46) TACR3TACR2OPRM1DHODHCYP2C9
Hydrochloric Acid SCHEMBL6953360 0.82 TACR3 (0.36) TACR3KCNH2GAATACR2OPRM1
SCHEMBL6586109 0.80 TRPV4 (0.43) TACR3KCNH2TACR2OPRM1DHODH
SCHEMBL6340547 0.80 TACR3 (0.40) TACR3KCNH2TACR2OPRM1DHODH
SCHEMBL7166157 0.80 DHODH (0.50) TACR3TACR2OPRM1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339691-A1 NOVEL COMPOUNDS GlaxoSmithKline S.p.A. (IT) 2003-09-03 EP disclosed
WO-2002044154-A1 NOVEL COMPOUNDS GLAXOSMITHKLINE SPA (IT) 2002-06-06 WO disclosed