SCHEMBL716423

SCHEMBL716423

O=C(O)CNC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCC(=O)N1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRHR P34981 5/20 0.41
HDAC3 O15379 4/20 0.37
HDAC11 Q96DB2 4/20 0.37
HDAC6 Q9UBN7 4/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC10 Q969S8 3/20 0.37
HDAC8 Q9BY41 3/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28309876 1.00 TRHR (0.41) TRHRHDAC3HDAC11HDAC6HDAC1
SCHEMBL11231582 1.00 TRHR (0.41) TRHRHDAC3HDAC11HDAC6HDAC1
SCHEMBL29405912 0.88 TRHR (0.46) TRHR
SCHEMBL27869228 0.88 TRHR (0.46) TRHR
SCHEMBL6026780 0.88 TRHR (0.46) TRHR
SCHEMBL6026783 0.88 TRHR (0.46) TRHR
SCHEMBL11034489 0.88 TRHR (0.44) TRHR
SCHEMBL3359034 0.85 TRHR (0.44) TRHR
SCHEMBL27209499 0.85 TRHR (0.56) TRHR
SCHEMBL8268065 0.85 TRHR (0.42) TRHRHDAC3HDAC11HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240075043-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2024-03-07 US claimed
US-20220249505-A1 APPETITE SUPPRESSANT COMPOSITIONS AND METHODS THEREOF RED MOUNTAIN HOLDINGS, LLC (US) 2022-08-11 US claimed
US-20210275536-A1 APPETITE SUPPRESSANT COMPOSITIONS AND METHODS THEREOF RED MOUNTAIN HOLDINGS, LLC (US) 2021-09-09 US claimed
WO-2009049105-A2 METHODS FOR INDUCING SATIATION GELESIS, INC. (US) 2009-04-16 WO claimed
EP-0394283-B1 USE OF A TRIPEPTIDE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS AND A PHARMACEUTICAL COMPOSITION AND METHOD Hafslund Nycomed AS (NO) 1992-12-02 EP claimed
EP-0394283-A1 USE OF A TRIPEPTIDE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS AND A PHARMACEUTICAL COMPOSITION AND METHOD. BIO TECH AS (NO) 1990-10-31 EP claimed
US-4956344-A PYROGLUTAMYLHISTIDYLGLYCINE ANTICARCINOGENIC AGENTS HAFSLUND NYCOMED A/S (NO) 1990-09-11 US claimed
WO-1989002276-A1 USE OF A TRIPEPTIDE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS AND A PHARMACEUTICAL COMPOSITION AND METHOD BIO-TECH A/S (NO) 1989-03-23 WO claimed
EP-0001174-B1 A PEPTIDE AND THE SALTS THEREOF, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM NYEGAARD & CO. A/S (NO) 1981-08-12 EP claimed
US-20250249016-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2025-08-07 US disclosed
US-20250249018-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS INCLUDING BUPROPION FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2025-08-07 US disclosed
US-20250249017-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS INCLUDING NALTREXONE FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2025-08-07 US disclosed
US-12303514-B2 Immediate and controlled release appetite suppressant compositions for weight loss Red Mountain Med Spa, LLC (US) 2025-05-20 US disclosed
US-20240075043-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2024-03-07 US disclosed
US-4956344-A PYROGLUTAMYLHISTIDYLGLYCINE ANTICARCINOGENIC AGENTS HAFSLUND NYCOMED A/S (NO) 1990-09-11 US disclosed
WO-1989002276-A1 USE OF A TRIPEPTIDE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS AND A PHARMACEUTICAL COMPOSITION AND METHOD BIO-TECH A/S (NO) 1989-03-23 WO disclosed
WO-1989002276-A1 USE OF A TRIPEPTIDE FOR THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS AND A PHARMACEUTICAL COMPOSITION AND METHOD BIO-TECH A/S (NO) 1989-03-23 WO disclosed
EP-0001174-B1 A PEPTIDE AND THE SALTS THEREOF, PROCESSES FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM NYEGAARD & CO. A/S (NO) 1981-08-12 EP disclosed
US-4260601-A PYROGLUTAMYL-HISTIDYL-GLYCINE, ANOREXIGENIC AGENT, IMMUNOASSAY/ KINSON*S DISEASE NYEGAARD & CO. A/S (NO) 1981-04-07 US disclosed
EP-0001174-A1 A peptide and the salts thereof, processes for their preparation and compositions containing them NYEGAARD & CO. A/S (NO) 1979-03-21 EP disclosed