SCHEMBL7164667

SCHEMBL7164667

COc1cc(OC)c(NC(=S)Nc2ccc(NC(=O)c3ccc(Cl)o3)cc2)cc1Cl

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.64
KMT2A Q03164 5/20 0.64
GAA P10253 3/20 0.64
NPSR1 Q6W5P4 2/20 0.64
MAPT P10636 9/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
ALDH1A1 P00352 8/20 0.57
HPGD P15428 3/20 0.57
LMNA P02545 2/20 0.57
KDM4E B2RXH2 5/20 0.53
HTT P42858 1/20 0.53
HSD17B10 Q99714 2/20 0.48
USP2 O75604 1/20 0.48
GRM4 Q14833 1/20 0.48
TSHR P16473 2/20 0.47
TAAR1 Q96RJ0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162969 0.92 MEN1 (0.78) MEN1KMT2AGAANPSR1MAPT
SCHEMBL7162179 0.84 KMT2A (0.54) MEN1KMT2AGAANPSR1MAPT
SCHEMBL7165683 0.83 MAPT (0.55) MEN1KMT2AGAANPSR1MAPT
SCHEMBL7163728 0.83 KDM4E (0.72) MEN1KMT2AGAANPSR1MAPT
SCHEMBL7165775 0.81 MAPT (0.67) MEN1KMT2AGAANPSR1MAPT
SCHEMBL6812142 0.81 MAPT (0.67) MEN1KMT2AGAANPSR1MAPT
SCHEMBL7939055 0.81 MAPT (0.70) MEN1KMT2AGAANPSR1MAPT
SCHEMBL6815648 0.81 MAPT (0.70) MEN1KMT2AGAANPSR1MAPT
SCHEMBL6815144 0.80 MAPT (0.62) MEN1KMT2AGAANPSR1MAPT
SCHEMBL6815565 0.80 MAPT (0.62) MEN1KMT2AGAANPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6555561-B2 N-(5-((((5-Chloro-2,4-dimethoxyphenyl)amino)thioxomethyl)-amino)-2 -pyridinyl)-2-methylbenzamide, for example; inhibiting replication of a herpes virus WYETH 2003-04-29 US disclosed