SCHEMBL7168254

SCHEMBL7168254

O=[N+]([O-])c1cc(F)ccc1OCC1CO1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPB1 P04792 3/20 0.45
ALDH1A1 P00352 4/20 0.44
GLA P06280 1/20 0.44
TDP1 Q9NUW8 2/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40
NPC1 O15118 1/20 0.40
RECQL P46063 1/20 0.40
RAB9A P51151 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3815074 0.90 TDP1 (0.47) HSPB1ALDH1A1GLATDP1ATM
SCHEMBL4824611 0.90 TDP1 (0.47) HSPB1ALDH1A1GLATDP1ATM
SCHEMBL1136179 0.86 TSHR (0.44) HSPB1ALDH1A1TSHRKMT2AMAPT
SCHEMBL30121999 0.84 MAPT (0.51) HSPB1ALDH1A1GLATDP1PRMT5
SCHEMBL3701823 0.84 MAPT (0.51) HSPB1ALDH1A1GLATDP1PRMT5
SCHEMBL9066974 0.83 KDM4E (0.51) ALDH1A1GLAL3MBTL1NPC1RAB9A
SCHEMBL1136235 0.83 HTR2A (0.51) HSPB1TDP1ATML3MBTL1NPC1
SCHEMBL4211452 0.82 NPC1 (0.60) ALDH1A1GLATDP1L3MBTL1NPC1
SCHEMBL4211458 0.82 NPC1 (0.60) ALDH1A1GLATDP1L3MBTL1NPC1
SCHEMBL3808783 0.82 NPC1 (0.60) ALDH1A1GLATDP1L3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6573377-B1 Antitumor agent capable of showing its efficacy even against 5- FU drug resistant tumors DAIICHI PHARMACEUTICALS CO., LTD. (JP) 2003-06-03 US disclosed
US-6552018-B1 As antitumor agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-22 US disclosed
EP-1103551-A1 PYRAZOLE DERIVATIVES AND SALTS THEREOF DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-05-30 EP disclosed
US-6169086-B1 AN ANTITUMOR AGENT FOR TREATING TUMOR RESISTANT TO 5-FLUOROURACIL TYPE DRUGS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-01-02 US disclosed