SCHEMBL7169286

SCHEMBL7169286

O=C(O)c1cncn1Cc1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 9/20 0.57
CYP11B2 P19099 9/20 0.57
GPBAR1 Q8TDU6 2/20 0.52
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
RAB9A P51151 1/20 0.44
IDO1 P14902 1/20 0.44
CNR2 P34972 1/20 0.44
GRM2 Q14416 1/20 0.43
CYP19A1 P11511 1/20 0.41
KDM4A O75164 1/20 0.41
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL753015 0.86 CYP11B1 (0.55) CYP11B1CYP11B2GPBAR1CA12CA1
SCHEMBL3932992 0.85 CYP11B1 (0.56) CYP11B1CYP11B2GPBAR1IDO1
SCHEMBL15795442 0.84 CYP11B1 (0.56) CYP11B1CYP11B2GPBAR1IDO1CYP19A1
Hydrochloric Acid SCHEMBL28186334 0.84 CYP11B1 (0.54) CYP11B1CYP11B2GPBAR1IDO1
SCHEMBL7488391 0.84 CYP11B1 (0.47) CYP11B1CYP11B2GPBAR1IDO1
SCHEMBL27353030 0.83 CYP11B1 (0.54) CYP11B1CYP11B2GPBAR1IDO1CYP19A1
SCHEMBL17684662 0.82 CYP11B1 (0.70) CYP11B1CYP11B2GPBAR1CA12CA1
SCHEMBL9121334 0.81 CYP11B1 (0.55) CYP11B1CYP11B2GPBAR1RAB9AIDO1
SCHEMBL9091320 0.81 CYP11B1 (0.54) CYP11B1CYP11B2GPBAR1RAB9AIDO1
SCHEMBL6708657 0.81 CYP11B1 (0.72) CYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083897-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-01-02 EP disclosed
EP-1083897-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-21 EP disclosed
WO-1999062513-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed