SCHEMBL7488391

SCHEMBL7488391

O=C(O)c1cncn1Cc1ccncc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 8/20 0.47
CYP11B2 P19099 7/20 0.47
GPBAR1 Q8TDU6 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CCNC P24863 1/20 0.43
CDK8 P49336 1/20 0.43
IDO1 P14902 1/20 0.42
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
MARS1 P56192 1/20 0.39
CNOT7 Q9UIV1 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3932992 0.88 CYP11B1 (0.56) CYP11B1CYP11B2GPBAR1CCNCCDK8
Hydrochloric Acid SCHEMBL28186334 0.87 CYP11B1 (0.54) CYP11B1CYP11B2GPBAR1CCNCCDK8
SCHEMBL15795442 0.84 CYP11B1 (0.56) CYP11B1CYP11B2GPBAR1IDO1PKM
SCHEMBL7169286 0.84 CYP11B1 (0.57) CYP11B1CYP11B2GPBAR1IDO1
SCHEMBL27353030 0.83 CYP11B1 (0.54) CYP11B1CYP11B2GPBAR1CCNCCDK8
SCHEMBL28683880 0.81 CYP11B1 (0.70) CYP11B1CYP11B2TSHRALDH1A1
SCHEMBL6708657 0.80 CYP11B1 (0.72) CYP11B1CYP11B2
SCHEMBL15654239 0.80 CCR9 (0.47) CYP11B1CYP11B2IDO1ALDH1A1MMP13
SCHEMBL7818410 0.79 CYP11B1 (0.70) CYP11B1CYP11B2
SCHEMBL26202128 0.77 CCR2 (0.53) CYP11B1CYP11B2GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196384-A4 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO INC (US) 2002-10-23 EP disclosed
EP-1196384-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF Merck & Co., Inc. (US) 2002-04-17 EP disclosed
WO-2001000578-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO., INC. (US) 2001-01-04 WO disclosed