SCHEMBL7170387

SCHEMBL7170387

COc1ccccc1Sc1ccc(C2CC2C(=O)NC(C)CC(=O)O)c(Cl)c1Cl

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 12/20 0.61
ICAM1 P05362 12/20 0.61
ITGAL P20701 12/20 0.61
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CHRNA7 P36544 1/20 0.36
GPR88 Q9GZN0 2/20 0.35
PLD2 O14939 1/20 0.33
PLD1 Q13393 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7170389 0.83 ITGB2 (0.75) ITGB2ICAM1ITGALKDM4ETDP1
SCHEMBL7143425 0.71 ITGAL (0.74) ITGB2ICAM1ITGAL
SCHEMBL7144870 0.69 ITGB2 (0.70) ITGB2ICAM1ITGAL
SCHEMBL2963974 0.65 CA1 (0.42) KDM4ETDP1
SCHEMBL6199566 0.65 ITGAL (0.51) ITGB2ICAM1ITGAL
SCHEMBL7147403 0.63 ITGB2 (0.50) ITGB2ICAM1ITGAL
SCHEMBL6792300 0.62 MMP2 (0.60) TDP1
SCHEMBL4278725 0.62 ITGAL (0.67) ITGB2ICAM1ITGALKDM4E
SCHEMBL4278719 0.62 ITGAL (0.67) ITGB2ICAM1ITGALKDM4E
Hydrogen Peroxide SCHEMBL28640288 0.62 CA1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521619-B2 Bind to the interaction-domain of integrin lfa-1 interrupting enothelial cell-leukocyte adhesion ICOS CORPORATION 2003-02-18 US claimed