SCHEMBL7174159

SCHEMBL7174159

Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2c(c1)c(-c1cccc(C#Cc3ccccc3)c1)cc(=O)n2C

nearest known ligand 0.80

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 9/20 0.80
FNTB P49356 9/20 0.80
CYP3A4 P08684 7/20 0.62
RORC P51449 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722541 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL12022163 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL5722562 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL7256220 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL4294372 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL12022161 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
SCHEMBL1643357 0.92 FNTA (0.78) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL4277842 0.91 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL30481066 0.91 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL21055098 0.91 FNTA (0.81) FNTAFNTBCYP3A4RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6579887-B2 Effective in inhibiting farnesyl protein transferase; also useful in treating benign proliferative disease. PFIZER INC 2003-06-17 US disclosed
US-20020128287-A1 Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents LYSSIKATOS JOSEPH P (US) 2002-09-12 US disclosed
US-6294552-B1 TREATMENT OF HYPERPROLIFERATIVE DISORDERS, SUCH AS CANCER, IN MAMMALS. THE INVENTION ALSO RELATES TO METHODS OF INHIBITING ABNORMAL CELL GROWTH, INCLUDING CANCER, IN A MAMMAL BY ADMINISTERING THE COMPOUNDS OF FORMULA 1 TO A MAMMAL REQUIRING PFIZER INC. 2001-09-25 US disclosed
US-6150377-A Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents PFIZER INC. (US) 2000-11-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020128287-A1 Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents CCNA1, NRAS, CCNT1 FNTA 1890/4885FNTB 2727/4885CYP3A4 1460/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.