Cp-609754

Cp-609754

SCHEMBL21055098

C#Cc1cccc(-c2cc(=O)n(C)c3ccc([C@](O)(c4ccc(Cl)cc4)c4cncn4C)cc23)c1

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 10/20 0.81
FNTB P49356 10/20 0.81
CYP3A4 P08684 8/20 0.59
RORC P51449 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cp-609754 SCHEMBL4277842 1.00 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL6583247 1.00 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL4299341 1.00 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL1644297 1.00 FNTA (0.81) FNTAFNTBCYP3A4RORC
Cp-609754 SCHEMBL30481066 1.00 FNTA (0.81) FNTAFNTBCYP3A4RORC
SCHEMBL11947163 0.93 FNTA (0.70) FNTAFNTBCYP3A4RORC
SCHEMBL12021644 0.93 FNTA (0.69) FNTAFNTBCYP3A4RORC
SCHEMBL13573622 0.92 FNTA (0.81) FNTAFNTBCYP3A4RORC
SCHEMBL11955976 0.92 FNTA (0.68) FNTAFNTBCYP3A4RORC
SCHEMBL11954234 0.91 FNTA (0.67) FNTAFNTBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230201183-A1 METHODS TO SYNERGISTICALLY ENHANCE MULTIPLE CELLULAR PROTEOSTASIS PATHWAYS TO TREAT NEURODEGENERATION AND STORAGE DISEASES NORTHWESTERN UNIVERSITY 2023-06-29 US disclosed
US-20230201183-A1 METHODS TO SYNERGISTICALLY ENHANCE MULTIPLE CELLULAR PROTEOSTASIS PATHWAYS TO TREAT NEURODEGENERATION AND STORAGE DISEASES NORTHWESTERN UNIVERSITY 2023-06-29 US disclosed
US-20230201183-A1 METHODS TO SYNERGISTICALLY ENHANCE MULTIPLE CELLULAR PROTEOSTASIS PATHWAYS TO TREAT NEURODEGENERATION AND STORAGE DISEASES NORTHWESTERN UNIVERSITY 2023-06-29 US disclosed
CN-114306604-A Use of farnesyl transferase inhibitors for the treatment of cancer 库拉肿瘤学公司 2022-04-12 CN disclosed
CN-110325212-B Farnesyl transferase inhibitors for use in methods of treating cancer 库拉肿瘤学公司 2022-03-22 CN disclosed
CN-114107497-A Use of farnesyl transferase inhibitors for the treatment of cancer 库拉肿瘤学公司 2022-03-01 CN disclosed
CN-111214658-B Methods of treating cancer patients with farnesyl transferase inhibitors 库拉肿瘤学公司 2022-01-11 CN disclosed
CN-107787373-B Use of farnesyl transferase inhibitors for the treatment of cancer 库拉肿瘤学公司 2021-11-26 CN disclosed
CN-111214658-A Methods of treating cancer patients with farnesyl transferase inhibitors 库拉肿瘤学公司 2020-06-02 CN disclosed
WO-2019113269-A1 METHODS OF TREATING CANCER PATIENTS WITH FARNESYLTRANSFERASE INHIBITORS KURA ONCOLOGY, INC. (US) 2019-06-13 WO disclosed
US-20100331363-A1 TREATMENT OF MITOCHONDRIAL DISORDERS USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-12-30 US disclosed
WO-2010057028-A9 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-09-02 WO disclosed
WO-2010056985-A9 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-08-19 WO disclosed
US-20100160372-A1 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-06-24 US disclosed
US-20100160372-A1 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-06-24 US disclosed
WO-2010057028-A2 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-05-20 WO disclosed
WO-2010056985-A2 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR LINK MEDICINE CORPORATION (US) 2010-05-20 WO disclosed
WO-2009151683-A2 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS LINK MEDICINE CORPORATION (US) 2009-12-17 WO disclosed
US-20090253655-A1 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS ASTRAZENECA AB (SE) 2009-10-08 US disclosed
US-20090253655-A1 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS ASTRAZENECA AB (SE) 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230201183-A1 METHODS TO SYNERGISTICALLY ENHANCE MULTIPLE CELLULAR PROTEOSTASIS PATHWAYS TO TREAT NEURODEGENERATION AND STORAGE DISEASES HSPA5, GBA1, SNCA FNTA 874/4885FNTB 1328/4885CYP3A4 4739/4885
US-20090253655-A1 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS PANK1, PANK3, PANK2 FNTA 4/4885FNTB 19/4885CYP3A4 3795/4885
US-20100160372-A1 TREATMENT OF PROTEINOPATHIES USING A FARNESYL TRANSFERASE INHIBITOR FNTA, FNTB, BDNF FNTA 1/4885FNTB 2/4885CYP3A4 3236/4885
US-20100331363-A1 TREATMENT OF MITOCHONDRIAL DISORDERS USING A FARNESYL TRANSFERASE INHIBITOR NLN, ACAT1, FH FNTA 7/4885FNTB 8/4885CYP3A4 1658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.