SCHEMBL7176261

SCHEMBL7176261

CC(=O)/C(=C\c1ccncc1)c1ccccc1.CC(=O)/C(=C\c1ccncc1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.58
CYP11B2 P19099 1/20 0.58
AKR1C1 Q04828 4/20 0.55
CYP1A2 P05177 4/20 0.50
CYP2D6 P10635 4/20 0.50
CYP2C9 P11712 4/20 0.50
CYP2C19 P33261 4/20 0.50
CYP3A4 P08684 3/20 0.50
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
AKR1C2 P52895 3/20 0.47
AKR1C3 P42330 2/20 0.47
HPGD P15428 5/20 0.47
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698550 1.00 CYP19A1 (0.58) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL6076208 1.00 CYP19A1 (0.58) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL7176266 1.00 CYP19A1 (0.58) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL5698547 1.00 CYP19A1 (0.58) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL5253679 0.93 AKR1C1 (0.55) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL5253681 0.93 AKR1C1 (0.55) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6
SCHEMBL6172379 0.87 AKR1C1 (0.70) AKR1C1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7992874 0.87 AKR1C1 (0.70) AKR1C1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5183481 0.87 AKR1C1 (0.70) AKR1C1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5698641 0.84 CYP19A1 (0.59) CYP19A1CYP11B2AKR1C1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6579873-B2 Treatment of inflammation, arthritis, bone disorders, respiratory system disorders PHARMACIA CORPORATION 2003-06-17 US disclosed