SCHEMBL718072

SCHEMBL718072

O=C1CCCC(=O)N1c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.63
MEN1 O00255 2/20 0.59
ALDH1A1 P00352 3/20 0.59
LMNA P02545 1/20 0.52
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA9 Q16790 1/20 0.50
MGLL Q99685 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
HPGD P15428 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HSD17B10 Q99714 1/20 0.47
MT-CO2 P00403 1/20 0.46
ALOX5 P09917 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23841260 0.95 KMT2A (0.65) KMT2AMEN1ALDH1A1LMNACA12
SCHEMBL370611 0.90 KMT2A (0.64) KMT2AMEN1ALDH1A1CA12CA1
SCHEMBL9073358 0.87 KMT2A (0.60) KMT2AMEN1ALDH1A1LMNACA12
SCHEMBL31068289 0.82 ALDH1A1 (0.61) KMT2AMEN1ALDH1A1MGLLL3MBTL1
SCHEMBL9627340 0.82 HPGD (0.66) KMT2AMEN1ALDH1A1LMNAHPGD
SCHEMBL12081988 0.80 MEN1 (0.64) KMT2AMEN1ALDH1A1MGLLHPGD
SCHEMBL22580612 0.80 MEN1 (0.64) KMT2AMEN1ALDH1A1MGLLHPGD
SCHEMBL12362822 0.79 MEN1 (0.57) KMT2AMEN1ALDH1A1MGLLHPGD
SCHEMBL29249691 0.79 KMT2A (0.54) KMT2AMEN1ALDH1A1CA12CA1
Toluene SCHEMBL16823388 0.78 KMT2A (0.50) KMT2AMEN1ALDH1A1LMNACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4702014-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING BRAF VIA UBIQUITIN PROTEOSOME PATHWAY Nurix Therapeutics, Inc. (US) 2026-03-04 EP claimed
WO-2024227104-A1 BIFUNCTIONAL COMPOUNDS FOR DEGRADING BRAF VIA UBIQUITIN PROTEOSOME PATHWAY NURIX THERAPEUTICS, INC. (US) 2024-10-31 WO claimed
CN-118667066-A Polymer, preparation method, binder, positive electrode sheet, secondary battery and electricity utilization device 宁德时代新能源科技股份有限公司 2024-09-20 CN claimed
EP-0666848-B1 SUBSTITUTED N-PHENYLGLUTARIMIDES AND N-PHENYLGLUTARIC ACID AMIDES, THEIR PREPARATION AND USE IN AGRICULTURE BASF AG (DE) 1998-12-30 EP claimed
US-5698494-A Substituted N-phenylglutarimides and N-phenylglutaramides, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 1997-12-16 US claimed
EP-0666848-A1 SUBSTITUTED N-PHENYLGLUTARIMIDES AND N-PHENYLGLUTARIC ACID AMIDES, THEIR PREPARATION AND USE IN AGRICULTURE BASF Aktiengesellschaft (DE) 1995-08-16 EP claimed
WO-1994010147-A1 SUBSTITUTED N-PHENYLGLUTARIMIDES AND N-PHENYLGLUTARIC ACID AMIDES, THEIR PREPARATION AND USE IN AGRICULTURE BASF AKTIENGESELLSCHAFT (DE) 1994-05-11 WO claimed
US-5223018-A Selective CIBA-GEIGY CORPORATION (US) 1993-06-29 US claimed
EP-0391847-A1 1-Phenyl-piperidine-2,4-dione with herbicidal activity CIBA-GEIGY AG (CH) 1990-10-10 EP claimed
EP-4661875-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS DEGRADERS OF MK2 KINASE Celgene Corporation (US) 2025-12-17 EP disclosed
EP-4648853-A1 TARGETED DEGRADATION OF VAV1 Monte Rosa Therapeutics AG (CH) 2025-11-19 EP disclosed
CN-120092003-A CDK protein degrading agents, pharmaceutical compositions and therapeutic uses 拜欧斯瑞克斯公司 2025-06-03 CN disclosed
EP-4524194-A1 RESIN COMPOSITION AND MOLDED OBJECT Kuraray Co., Ltd. (JP) 2025-03-19 EP disclosed
CN-119343403-A Resin composition and molded article 株式会社可乐丽 2025-01-21 CN disclosed
US-3959286-A ANTIDEPRESSANTS, ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1976-05-25 US disclosed
US-3947452-A ANTIDEPRESSANT, ANTIANXIETY, ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1976-03-30 US disclosed
US-3940398-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1976-02-24 US disclosed
US-3940397-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1976-02-24 US disclosed
US-3935227-A ANTIDEPRESSANTS, ANTIANXIETY, ANTIINFLAMMATORY AGENTS E. R. SQUIBB & SONS, INC. (US) 1976-01-27 US disclosed
US-3933831-A Perfluorinated tertiary amines PCR, INC. (US) 1976-01-20 US disclosed