SCHEMBL7180720

SCHEMBL7180720

COC(=O)[C@H](Cc1ccc(N(C)c2ccncc2)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.54
RAB9A P51151 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
ITGB1 P05556 3/20 0.46
ITGA5 P08648 2/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
USP2 O75604 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
FKBP1A P62942 1/20 0.45
MAPT P10636 1/20 0.44
POLB P06746 1/20 0.44
KCNQ1 P51787 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7180590 0.92 ITGA4 (0.59) ITGA4GAAHPGDITGB1ITGA5
SCHEMBL7327448 0.86 ITGA4 (0.54) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL3849601 0.85 ITGA4 (0.60) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL6712426 0.85 ITGA4 (0.59) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL6709486 0.85 ITGA4 (0.59) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL5690332 0.85 ITGA4 (0.59) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL6709270 0.84 ITGA4 (0.60) ITGA4RAB9AGAAHPGDITGB1
SCHEMBL5690625 0.84 MAPK1 (0.66) ITGA4GAAITGB1ITGA5TSHR
SCHEMBL6710835 0.84 ITGA4 (0.55) ITGA4RAB9AITGB1ITGA5TSHR
SCHEMBL3850808 0.84 ITGA4 (0.55) ITGA4RAB9AGAAHPGDITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583139-B1 Treatment of inflammatory diseases; inflammatory brain diseases such as multiple sclerosis; N-(Toluene-4-sulfonyl)-L-prolyl-4-(alpha -methylbenzyloxy)-L-phenylalanine; Very Late Antigen 4 BIOGEN IDEC INTERNATIONAL HOLDING LTD. (BM) 2003-06-24 US disclosed