SCHEMBL7181653

SCHEMBL7181653

CCc1cc2c(Cl)nc(CCCCCCC(=O)OC)nc2s1.CCc1cc2c(NCc3ccc4c(c3)OCO4)nc(CCCCCCC(=O)OC)nc2s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
PPP1CA P62136 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RAB9A P51151 1/20 0.38
PDE5A O76074 4/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PDE2A O00408 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6707067 0.95 ALDH1A1 (0.42) SMN1; SMN2ALDH1A1HTTKDM4EPOLB
SCHEMBL6707030 0.95 ALDH1A1 (0.42) SMN1; SMN2ALDH1A1HTTKDM4EPOLB
SCHEMBL7099400 0.92 SMN1; SMN2 (0.40) SMN1; SMN2ALDH1A1KDM4EPOLBMAPT
SCHEMBL6709515 0.92 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1HTTKDM4EPOLB
SCHEMBL7095239 0.92 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1KDM4EPOLBMAPT
SCHEMBL6709505 0.89 HDAC3 (0.41) SMN1; SMN2ALDH1A1KDM4EPOLBMAPT
SCHEMBL6706987 0.89 ALDH1A1 (0.44) SMN1; SMN2ALDH1A1HTTKDM4EPOLB
SCHEMBL6709592 0.88 HSD17B10 (0.41) SMN1; SMN2ALDH1A1KDM4EPOLBMAPT
SCHEMBL6709541 0.88 KDM4E (0.46) SMN1; SMN2ALDH1A1HTTKDM4EPOLB
SCHEMBL6763990 0.87 KDM4E (0.46) SMN1; SMN2ALDH1A1HTTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355649-A2 PHARMACEUTICAL FORMULATION CONTAINING PYRAZOLO 4,3-D]PYRIMIDINE AND NITRATES OR THIENOPYRIMIDINES AND NITRATES MERCK PATENT GmbH (DE) 2003-10-29 EP disclosed
WO-2002060449-A2 PHARMACEUTICAL FORMULATION CONTAINING PYRAZOLO[4,3-D]PYRIMIDINE AND NITRATES OR THIENOPYRIMIDINES AND NITRATES MERCK PATENT GMBH (DE) 2002-08-08 WO disclosed