SCHEMBL7182779

SCHEMBL7182779

CCOC(=O)C=Cc1ccc(Oc2c(-c3ccc(Cl)cc3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.52
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
ESR2 Q92731 7/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7188067 0.94 CA12 (0.56) ESR1CA12CA1CA2CA7
SCHEMBL7192245 0.92 CYP3A4 (0.48) ESR1CA12CA1CA2CA7
SCHEMBL7191463 0.91 ESR1 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL7186125 0.88 ESR1 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL7183887 0.86 ESR1 (0.54) ESR1CA12CA1CA2CA7
SCHEMBL7189967 0.86 ESR1 (0.64) ESR1ESR2
SCHEMBL7189970 0.86 ESR1 (0.64) ESR1ESR2
SCHEMBL7182803 0.86 ESR1 (0.54) ESR1ESR2
SCHEMBL7184090 0.85 CYP3A4 (0.52) ESR1CA12CA1CA2CA7
SCHEMBL7193933 0.85 ESR1 (0.54) ESR1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP claimed