SCHEMBL7185591

SCHEMBL7185591

COc1cc(CC=C(C)C)ccc1C=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
PTGS1 P23219 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TDP1 Q9NUW8 2/20 0.44
KDM4E B2RXH2 2/20 0.44
TSHR P16473 1/20 0.44
CYP3A4 P08684 2/20 0.43
ALOX5 P09917 1/20 0.43
AR P10275 1/20 0.43
TRPM8 Q7Z2W7 1/20 0.43
ERN1 O75460 3/20 0.43
PPARG P37231 1/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
TLR2 O60603 1/20 0.42
TLR1 Q15399 1/20 0.42
TLR6 Q9Y2C9 1/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15156353 0.81 ALDH1A1 (0.67) ALDH1A1PTGS1L3MBTL1TDP1KDM4E
SCHEMBL14447279 0.80 ALDH1A1 (0.58) ALDH1A1PTGS1L3MBTL1TDP1KDM4E
SCHEMBL10908228 0.79 ALDH1A1 (0.68) ALDH1A1PTGS1TDP1TSHRCYP3A4
SCHEMBL9714792 0.78 ALDH1A1 (0.59) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL14327024 0.77 ALDH1A1 (0.58) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL28783867 0.77 ALDH1A1 (0.58) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL29956536 0.76 ALDH1A1 (0.64) ALDH1A1PTGS1L3MBTL1TDP1KDM4E
SCHEMBL7179024 0.76 ALDH1A1 (0.61) ALDH1A1L3MBTL1KDM4EALOX5MAPT
SCHEMBL465084 0.76 ALDH1A1 (0.56) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL9958482 0.76 HTT (0.41) ALDH1A1PTGS1CYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed