SCHEMBL7185985

SCHEMBL7185985

CCCOc1cc(O)c(C)cc1/C=C/C(=O)c1ccc(N)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.56
DPP4 P27487 8/20 0.55
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.46
AR P10275 1/20 0.45
CYP1A1 P04798 1/20 0.44
CYP1B1 Q16678 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185991 1.00 PTPN1 (0.56) PTPN1DPP4CTSLCTSBABCG2
SCHEMBL7189383 0.91 PTPN1 (0.58) PTPN1DPP4CTSLCTSBCA1
SCHEMBL7187836 0.91 DPP4 (0.57) PTPN1DPP4CTSLCTSBABCG2
SCHEMBL7187835 0.91 DPP4 (0.57) PTPN1DPP4CTSLCTSBABCG2
SCHEMBL7189381 0.91 PTPN1 (0.58) PTPN1DPP4CTSLCTSBCA1
SCHEMBL7182974 0.91 DPP4 (0.49) PTPN1DPP4CTSLCTSBABCG2
SCHEMBL7184832 0.89 PTPN1 (0.56) PTPN1DPP4CTSLCTSB
SCHEMBL7184838 0.89 PTPN1 (0.56) PTPN1DPP4CTSLCTSB
SCHEMBL7184454 0.87 PTPN1 (0.54) PTPN1DPP4CTSLCTSB
SCHEMBL7184456 0.87 PTPN1 (0.54) PTPN1DPP4CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed