SCHEMBL7187835

SCHEMBL7187835

CCCOc1cc(O)c(C)cc1/C=C/C(=O)c1ccc(O)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 10/20 0.57
ABCG2 Q9UNQ0 3/20 0.56
PTPN1 P18031 5/20 0.54
CAPN1 P07384 1/20 0.53
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CHRNA7 P36544 1/20 0.49
IDH1 O75874 1/20 0.48
ABCB1 P08183 1/20 0.48
UGT1A1 P22309 1/20 0.48
ABCC1 P33527 1/20 0.48
PRMT6 Q96LA8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7187836 1.00 DPP4 (0.57) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL9204823 0.94 PTPN1 (0.55) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL9204820 0.94 PTPN1 (0.55) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL7180998 0.92 ABCG2 (0.57) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL7185991 0.91 PTPN1 (0.56) DPP4ABCG2PTPN1CTSLCTSB
SCHEMBL7185985 0.91 PTPN1 (0.56) DPP4ABCG2PTPN1CTSLCTSB
SCHEMBL7185020 0.90 DPP4 (0.56) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL7185017 0.90 DPP4 (0.56) DPP4ABCG2PTPN1CAPN1CTSL
SCHEMBL7192343 0.89 DPP4 (0.53) DPP4ABCG2PTPN1
SCHEMBL7192340 0.89 DPP4 (0.53) DPP4ABCG2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed