SCHEMBL7186727

SCHEMBL7186727

C=CCOc1ccc(C(=O)C=Cc2c(OCCCC)cccc2OCCCC)cc1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.52
PTPN1 P18031 2/20 0.49
BCHE P06276 10/20 0.49
ACHE P22303 8/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
DPP4 P27487 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7179229 0.95 ABCG2 (0.52) ABCG2PTPN1BCHEACHECHRNB2
SCHEMBL7186353 0.91 MAOB (0.54) ABCG2PTPN1MAOAMAOB
SCHEMBL7182892 0.91 MAOB (0.54) ABCG2PTPN1MAOAMAOB
SCHEMBL7184568 0.87 ABCG2 (0.70) ABCG2PTPN1MAOAMAOB
SCHEMBL7184561 0.87 ABCG2 (0.70) ABCG2PTPN1MAOAMAOB
SCHEMBL7183784 0.87 ABCG2 (0.48) ABCG2PTPN1BCHEACHEMAOA
SCHEMBL7803247 0.85 ABCG2 (0.52) ABCG2PTPN1CHRNB2CHRNB4CHRNA3
SCHEMBL7191615 0.85 ABCG2 (0.52) ABCG2PTPN1CHRNB2CHRNB4CHRNA3
SCHEMBL7184476 0.84 ABCG2 (0.64) ABCG2PTPN1BCHEACHEMAOB
SCHEMBL7184195 0.84 PTPN1 (0.46) ABCG2PTPN1BCHEACHEDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US claimed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP claimed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP claimed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO claimed