SCHEMBL7186899

SCHEMBL7186899

CC(C)Oc1cccc(OC(C)C)c1/C=C/C(=O)c1ccc(O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.61
MAOB P27338 2/20 0.55
MAPT P10636 3/20 0.50
KMT2A Q03164 2/20 0.50
MDM4 O15151 1/20 0.50
MDM2 Q00987 1/20 0.50
CAPN1 P07384 3/20 0.49
CTSL P07711 3/20 0.49
CTSB P07858 3/20 0.49
F3 P13726 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH2 P05091 1/20 0.49
CYP3A4 P08684 1/20 0.49
HSPD1 P10809 1/20 0.49
CYP19A1 P11511 1/20 0.49
MAOA P21397 1/20 0.49
HSPE1 P61604 1/20 0.49
CYP1B1 Q16678 1/20 0.49
P4HB P07237 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7186903 1.00 ABCG2 (0.61) ABCG2MAOBMAPTKMT2AMDM4
SCHEMBL7187753 0.87 ABCG2 (0.60) ABCG2MAOBMAPTKMT2ACTSL
SCHEMBL7187758 0.87 ABCG2 (0.60) ABCG2MAOBMAPTKMT2ACTSL
SCHEMBL7189354 0.85 ABCG2 (0.57) ABCG2MAOBMAPTCYP3A4MAOA
SCHEMBL7189351 0.85 ABCG2 (0.57) ABCG2MAOBMAPTCYP3A4MAOA
SCHEMBL7180373 0.85 ABCG2 (0.57) ABCG2MAOBMAPTKMT2AMAOA
SCHEMBL7180369 0.85 ABCG2 (0.57) ABCG2MAOBMAPTKMT2AMAOA
SCHEMBL7190678 0.84 CAPN1 (0.47) ABCG2MAOBMAPTKMT2ACAPN1
SCHEMBL7190676 0.84 CAPN1 (0.47) ABCG2MAOBMAPTKMT2ACAPN1
SCHEMBL7185747 0.84 ABCG2 (0.88) ABCG2MAOBMAPTKMT2ACAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed