SCHEMBL718949

SCHEMBL718949

Fc1ccc(C#Cc2ccc(F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.50
FFAR1 O14842 1/20 0.50
APP P05067 4/20 0.47
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA7 P43166 1/20 0.42
ACHE P22303 1/20 0.42
KDM4E B2RXH2 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
CA12 O43570 1/20 0.38
HAO1 Q9UJM8 1/20 0.37
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717366 1.00 GRM5 (0.50) GRM5FFAR1APPCA1CA2
SCHEMBL10300106 1.00 GRM5 (0.50) GRM5FFAR1APPCA1CA2
Fluoride SCHEMBL31286313 0.97 GRM5 (0.48) GRM5FFAR1APPCA1CA2
Charcoal, Activated SCHEMBL31286307 0.97 GRM5 (0.48) GRM5FFAR1APPCA1CA2
SCHEMBL13810534 0.91 GRM5 (0.45) GRM5FFAR1APPCA1CA2
SCHEMBL20212084 0.91 GRM5 (0.50) GRM5FFAR1APPCA1CA2
SCHEMBL18867945 0.88 APP (0.67) GRM5FFAR1APPCA1CA2
SCHEMBL717468 0.88 APP (0.67) GRM5FFAR1APPCA1CA2
SCHEMBL949444 0.86 APP (0.58) GRM5FFAR1APPCA1CA2
SCHEMBL8623669 0.86 SMN1; SMN2 (0.43) GRM5FFAR1APPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119661581-A Fused ring tin porphyrin photosensitizer with high singlet oxygen sensitization efficiency and photothermal effect 四川大学华西医院 2025-03-21 CN claimed
CN-119118977-A Preparation method of gamma-pyrone compound 西北工业大学 2024-12-13 CN claimed
CN-114560761-B Method for one-time synthesis of 2,3-disubstituted indanone derivative in aqueous phase 南京林业大学 2023-02-24 CN claimed
US-6761975-B1 RESISTANCE TO DELAMINATION; ELIMINATES THE NEED FOR A PRIMER COATING APPLICATION PROCESS STEP; CURABLE POLYARYL ETHER FILM HONEYWELL INTERNATIONAL INC. 2004-07-13 US claimed
US-20020198353-A1 Polycarbosilane adhesion promoters for low dielectric constant polymeric materials HONEYWELL INTERNATIONAL INC. 2002-12-26 US claimed
EP-1243003-A1 POLYCARBOSILANE ADHESION PROMOTERS FOR LOW DIELECTRIC CONSTANT POLYMERIC MATERIALS AlliedSignal Inc. (US) 2002-09-25 EP claimed
US-6380347-B1 MACROCYCLES MADE BY THE CYCLIZATION OF A BISPHENOL CONTAINING TRIPLE BOND(S) AND A DIFLUOROAROMATIC COMPOUND; MODIFIERS OF CROSSLINKED POLYMERS; LOW DIELECTRIC CONSTANT FOR THE LAYERS OF INTEGRATED CIRCUITS CONTAINING METALLIC CONNECTORS HONEYWELL INTERNATIONAL INC. 2002-04-30 US claimed
WO-2001046963-A1 POLYCARBOSILANE ADHESION PROMOTERS FOR LOW DIELECTRIC CONSTANT POLYMERIC MATERIALS ALLIEDSIGNAL INC. (US) 2001-06-28 WO claimed
US-6124421-A A SEMICONDUCTOR DEVICE COMPRISING A DIELECTRIC LAYER DISPOSED OVERLYING A SURFACE, COMPRISES A POLY(ARYLENE ETHER) ALLIEDSIGNAL INC. (US) 2000-09-26 US claimed
CN-119661581-A Fused ring tin porphyrin photosensitizer with high singlet oxygen sensitization efficiency and photothermal effect 四川大学华西医院 2025-03-21 CN disclosed
CN-119346167-A Catalytic system and method for synthesizing diaryl acetylene from calcium carbide and iodo aromatic hydrocarbon 石河子大学 2025-01-24 CN disclosed
CN-119118977-A Preparation method of gamma-pyrone compound 西北工业大学 2024-12-13 CN disclosed
CN-119019450-A Synthesis method of trisubstituted olefin carbazole phosphine ligand derivative 广西大学 2024-11-26 CN disclosed
CN-118420533-A Method for synthesizing isoquinolinone by carbonylation of aryl alkyne and hydroxylamine 中国科学技术大学 2024-08-02 CN disclosed
EP-1068255-A2 POLY(ARYLENE ETHER) COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF AlliedSignal Inc. (US) 2001-01-17 EP disclosed
US-6124421-A A SEMICONDUCTOR DEVICE COMPRISING A DIELECTRIC LAYER DISPOSED OVERLYING A SURFACE, COMPRISES A POLY(ARYLENE ETHER) ALLIEDSIGNAL INC. (US) 2000-09-26 US disclosed
WO-1999029761-A2 POLY(ARYLENE ETHER) COMPOSITIONS AND METHODS OF MANUFACTURE THEREOF ALLIEDSIGNAL INC. (US) 1999-06-17 WO disclosed
US-5374701-A Crosslinkable polymers of high strength free of structural defects HAY ALLAN S (CA) 1994-12-20 US disclosed
US-5233046-A DIARYLACETYLENES, ENAMINES AND ACETYLENIC POLYMERS AND THEIR PRODUCTION HAY ALLAN S (CA) 1993-08-03 US disclosed
WO-1993009079-A1 DIARYLACETYLENES, ENAMINES AND ACETYLENIC POLYMERS AND THEIR PRODUCTION HAY ALAN S (CA) 1993-05-13 WO disclosed