SCHEMBL7195077

SCHEMBL7195077

N#C/C(C(=O)O)=C(/C#N)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
XBP1 P17861 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HPGD P15428 2/20 0.30
CISD1 Q9NZ45 1/20 0.30
KDM4E B2RXH2 1/20 0.30
SLC16A3 O15427 1/20 0.30
CYP3A4 P08684 1/20 0.30
SLC16A1 P53985 1/20 0.30
GPR35 Q9HC97 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195083 1.00 ALDH1A1 (0.32) ALDH1A1MAPTLMNAXBP1MAPK1
SCHEMBL6924823 0.83
SCHEMBL16043962 0.83
SCHEMBL16043961 0.83
SCHEMBL1437550 0.81
SCHEMBL4507423 0.81
SCHEMBL4507427 0.81
SCHEMBL11006695 0.81
SCHEMBL4507425 0.81
SCHEMBL12669264 0.81 DHODH (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883652-B1 RADIATION CURABLE COATING COMPOSITION DSM NV (NL) 2000-03-15 EP claimed
US-6025409-A COMPRISING (A) UNSATURATED COMPOUND HAVING AT LEAST ONE MALEATE, FUMERATE, ITACONATE, CITRACONATE OR MESACONATE GROUP; (B) AN UNSATURATED VINYLETHER COMPOUND AND A COMPOUND WHICH FORMS A STRONG EXCIPLEX WITH (A) OR (B); DSM N.V. (NL) 2000-02-15 US claimed
EP-0883652-A1 RADIATION CURABLE COATING COMPOSITION DSM N.V. (NL) 1998-12-16 EP claimed
WO-1997031981-A1 RADIATION CURABLE COATING COMPOSITION DSM N.V. (NL) 1997-09-04 WO claimed
US-4535042-A Electrophotographic photosensitive member with electron donor and acceptor layers CANON KABUSHIKI KAISHA, A CORP. OF JAPAN (JP) 1985-08-13 US claimed
US-4225648-A PROTECTIVE COATING OF POLYMER CONTAINING LEWIS ACID RICOH COMPANY, LTD. (JP) 1980-09-30 US claimed
US-10309927-B2 Methods of conducting biochemical reactions while reducing reactive molecular species during electrowetting ILLUMINA, INC. (US) 2019-06-04 US disclosed
EP-3280819-B1 METHODS OF CONDUCTING BIOCHEMICAL REACTIONS WHILE REDUCING REACTIVE MOLECULAR SPECIES DURING ELECTROWETTING ILLUMINA INC (US) 2019-05-22 EP disclosed
EP-3280819-A1 METHODS OF CONDUCTING BIOCHEMICAL REACTIONS WHILE REDUCING REACTIVE MOLECULAR SPECIES DURING ELECTROWETTING Illumina, Inc. (US) 2018-02-14 EP disclosed
US-20160299101-A1 METHODS OF CONDUCTING BIOCHEMICAL REACTIONS WHILE REDUCING REACTIVE MOLECULAR SPECIES DURING ELECTROWETTING ILLUMINA, INC. 2016-10-13 US disclosed
WO-2016164592-A1 METHODS OF CONDUCTING BIOCHEMICAL REACTIONS WHILE REDUCING REACTIVE MOLECULAR SPECIES DURING ELECTROWETTING ILLUMINA, INC. (US) 2016-10-13 WO disclosed
US-6562181-B2 Bonding together two substrates by applying to a first substrate formulation of mixture of trifunctional olefinic monomer, olefinic second monomer that is copolymerizable and free radical initiator; contacting second substrate LORD CORPORATION 2003-05-13 US disclosed
US-20020129896-A1 REACTIVE ADHESIVES AND COATINGS WITH TRIFUNCTIONAL OLEFINIC MONOMERS LORD CORPORATION 2002-09-19 US disclosed
US-6025409-A COMPRISING (A) UNSATURATED COMPOUND HAVING AT LEAST ONE MALEATE, FUMERATE, ITACONATE, CITRACONATE OR MESACONATE GROUP; (B) AN UNSATURATED VINYLETHER COMPOUND AND A COMPOUND WHICH FORMS A STRONG EXCIPLEX WITH (A) OR (B); DSM N.V. (NL) 2000-02-15 US disclosed
WO-2000006613-A1 PHOTOPOLYMERIZATION PROCESS AND COMPOSITION EMPLOYING A CHARGE TRANSFER COMPLEX AND CATIONIC PHOTOINITIATOR FUSION UV SYSTEMS, INC. (US) 2000-02-10 WO disclosed
EP-0883652-A1 RADIATION CURABLE COATING COMPOSITION DSM N.V. (NL) 1998-12-16 EP disclosed
WO-1997031981-A1 RADIATION CURABLE COATING COMPOSITION DSM N.V. (NL) 1997-09-04 WO disclosed
US-4535042-A Electrophotographic photosensitive member with electron donor and acceptor layers CANON KABUSHIKI KAISHA, A CORP. OF JAPAN (JP) 1985-08-13 US disclosed
US-4469771-A POLYMERIC PROTECTIVE COATING CONTAINING LEWIS ACID RICOH CO., LTD. (JP) 1984-09-04 US disclosed
US-4225648-A PROTECTIVE COATING OF POLYMER CONTAINING LEWIS ACID RICOH COMPANY, LTD. (JP) 1980-09-30 US disclosed