SCHEMBL7201932

SCHEMBL7201932

NC(=O)c1ccnc(-c2ccccc2)c1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.46
MAP2K1 Q02750 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
CDC7 O00311 8/20 0.43
RXFP1 Q9HBX9 1/20 0.42
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
IKBKB O14920 3/20 0.41
PARP1 P09874 2/20 0.41
CDK2 P24941 3/20 0.41
CCNA2 P20248 2/20 0.41
CCNE1 P24864 2/20 0.41
CCNA1 P78396 2/20 0.41
CCNT1 O60563 1/20 0.41
JAK2 O60674 1/20 0.41
CCNB2 O95067 1/20 0.41
CCNE2 O96020 1/20 0.41
PRKCB P05771 1/20 0.41
CDK1 P06493 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217185 0.83 CDC7 (0.46) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL1758364 0.83 IKBKB (0.47) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL27890738 0.81 KDM4E (0.46) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL30096560 0.80 IKBKB (0.46) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL21626163 0.79 MAP2K1 (0.43) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL29916420 0.79 KDM4E (0.55) BCAT2MAP2K1CLK4DYRK1BKDM4E
SCHEMBL945856 0.79 KDM4E (0.55) BCAT2MAP2K1CLK4DYRK1BKDM4E
SCHEMBL27872332 0.76 MAP2K1 (0.41) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL21626162 0.76 MAP2K1 (0.43) BCAT2MAP2K1CLK4DYRK1BCDC7
SCHEMBL28941125 0.75 MAP2K1 (0.40) BCAT2MAP2K1CLK4DYRK1BCDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366016-A2 PROCESS FOR THE PREPARATION OF ARYLETHANOLDIAMINES USEFUL AS AGONISTS OF THE BETA-3-ADRENOCEPTOR GLAXO GROUP LIMITED (GB) 2003-12-03 EP disclosed
WO-2002066418-A2 PROCESS FOR THE PREPARATION OF ARYLETHANOLDIAMINES USEFUL AS AGONISTS OF THE BETA-3-ADRENOCEPTOR GLAXO GROUP LIMITED (GB) 2002-08-29 WO disclosed