SCHEMBL7203487

SCHEMBL7203487

[2H][C@H]1C(=O)[C@]([2H])(NC(=O)[CH]CC(C)C(N)=O)CCCN1S(=O)(=O)c1cccc[n+]1[O-]

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.40
PKM P14618 1/20 0.32
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6593103 1.00 CTSK (0.40) CTSKPKMDRD4
SCHEMBL5575176 0.94 CTSK (0.40) CTSKPKM
SCHEMBL6899315 0.92 CTSK (0.41) CTSKPKMDRD4
SCHEMBL4687353 0.85 CTSK (0.52) CTSKPKMDRD4
SCHEMBL5096677 0.85 CTSK (0.52) CTSKPKMDRD4
SCHEMBL4687256 0.82 CTSK (0.38) CTSKPKM
SCHEMBL4686550 0.82 CTSK (0.43) CTSK
SCHEMBL5949076 0.77 CTSK (0.33) CTSKPKM
SCHEMBL4686403 0.77 CTSK (0.54) CTSKPKMDRD4
SCHEMBL4315397 0.76 CTSK (0.38) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1229911-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-05-07 EP disclosed
EP-1229911-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2002-08-14 EP disclosed
WO-2001034153-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-17 WO disclosed