SCHEMBL7204268

SCHEMBL7204268

CCc1cccc(N(C)C(=N)N(C)c2cc(Br)ccc2Br)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 1.00
TP53 P04637 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
THPO P40225 1/20 0.41
MTOR P42345 1/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
PMP22 Q01453 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7206171 0.99 SIGMAR1 (1.00) SIGMAR1MEN1LMNAMAPTPMP22
SCHEMBL7070370 0.92 SIGMAR1 (0.85) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7206334 0.84 SIGMAR1 (0.73) SIGMAR1
SCHEMBL6722611 0.84 SIGMAR1 (0.73) SIGMAR1
SCHEMBL6720958 0.83 SIGMAR1 (0.73) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL7203955 0.82 SIGMAR1 (0.69) SIGMAR1
SCHEMBL6727640 0.78 SIGMAR1 (0.63) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6720673 0.78 SIGMAR1 (0.63) SIGMAR1LMNAMAPTKMT2A
SCHEMBL7647473 0.77 SIGMAR1 (0.74) SIGMAR1TP53CYP2D6TSHRTHPO
Hydrochloric Acid SCHEMBL7204073 0.77 SIGMAR1 (0.64) SIGMAR1MEN1LMNAMAPTPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705100-B1 THERAPEUTIC SUBSTITUTED GUANIDINES CENES LTD (GB) 2003-07-30 EP disclosed
US-6156741-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-12-05 US disclosed
US-6153604-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-11-28 US disclosed
US-6147063-A NEUROTOXICITY CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-11-14 US disclosed
EP-0705100-A4 THERAPEUTIC SUBSTITUTED GUANIDINES CAMBRIDGE NEUROSCIENCE INC (US) 1996-05-29 EP disclosed
EP-0705100-A1 THERAPEUTIC SUBSTITUTED GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1996-04-10 EP disclosed
WO-1994027591-A1 THERAPEUTIC SUBSTITUTED GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1994-12-08 WO disclosed