SCHEMBL7204503

SCHEMBL7204503

CC(=Cc1c(C(C)c2cc(C(C)(C)C)cc(C(C)(C)C)c2C=C(C)C(=O)O)cc(C(C)(C)C)cc1C(C)(C)C)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
RXRA P19793 9/20 0.33
PPARG P37231 8/20 0.33
AKR1C3 P42330 1/20 0.33
RARG P13631 3/20 0.33
ALOX5 P09917 1/20 0.31
PTGS2 P35354 1/20 0.31
RXRB P28702 3/20 0.31
RXRG P48443 3/20 0.31
TBXAS1 P24557 2/20 0.31
RARA P10276 2/20 0.31
RARB P10826 2/20 0.31
APEX1 P27695 1/20 0.31
GABBR2 O75899 1/20 0.31
GABBR1 Q9UBS5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL809465 0.94 CYP3A4 (0.43) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL809466 0.94 CYP3A4 (0.43) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL7205602 0.86 SMN1; SMN2 (0.36) CYP2C9CYP2C19AKR1C3TBXAS1APEX1
SCHEMBL7206085 0.82 HSPA5 (0.36) CYP1A2CYP3A4TSHRAKR1C3RARB
SCHEMBL7200632 0.81 RXRA (0.38) RXRAPPARGAKR1C3RARGRXRB
SCHEMBL7200672 0.78 CYP3A4 (0.37) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4145596 0.76 RXRA (0.35) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4145601 0.76 RXRA (0.35) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL14673352 0.73 HSPA5 (0.43) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL809386 0.73 CYP1A2 (0.44) CYP1A2CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028731-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed
US-6525120-B2 Stabilization using bisphenol ester SUMITOMO CHEMICAL CO., LTD. (JP) 2003-02-25 US disclosed
US-20020002249-A1 Polymer composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-01-03 US disclosed