SCHEMBL7204837

SCHEMBL7204837

CCc1cccc(N(C)C(N)=Nc2cc(C(F)(F)F)ccc2Br)c1

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.73
TP53 P04637 1/20 0.56
CYP2D6 P10635 1/20 0.56
TSHR P16473 1/20 0.56
THPO P40225 1/20 0.56
MTOR P42345 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7207724 0.99 SIGMAR1 (0.74) SIGMAR1
SCHEMBL6716544 0.91 SIGMAR1 (0.64) SIGMAR1
Hydrochloric Acid SCHEMBL7202394 0.90 SIGMAR1 (0.66) SIGMAR1
SCHEMBL7205171 0.88 SIGMAR1 (0.72) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6717076 0.87 SIGMAR1 (0.80) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6719635 0.87 SIGMAR1 (0.74) SIGMAR1
Hydrochloric Acid SCHEMBL7201854 0.87 SIGMAR1 (0.74) SIGMAR1
Hydrochloric Acid SCHEMBL7205189 0.86 SIGMAR1 (0.82) SIGMAR1
Hydrochloric Acid SCHEMBL7210031 0.86 SIGMAR1 (0.74) SIGMAR1
SCHEMBL6727642 0.85 SIGMAR1 (0.76) SIGMAR1TP53CYP2D6TSHRTHPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705100-B1 THERAPEUTIC SUBSTITUTED GUANIDINES CENES LTD (GB) 2003-07-30 EP claimed
US-6156741-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-12-05 US claimed
US-6153604-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-11-28 US claimed
US-6147063-A NEUROTOXICITY CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-11-14 US claimed
EP-0705100-B1 THERAPEUTIC SUBSTITUTED GUANIDINES CENES LTD (GB) 2003-07-30 EP disclosed
US-6153604-A Therapeutic substituted guanidines CAMBRIDGE NEUROSCIENCE, INC. (US) 2000-11-28 US disclosed