SCHEMBL7204850

SCHEMBL7204850

CCCCCCNCCCCCCO[C@H]1CC[C@H](N(C)C(=O)Cc2ccc(F)cc2F)CC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.42
LSS P48449 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
KCNH2 Q12809 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
DPP4 P27487 3/20 0.36
DPP9 Q86TI2 2/20 0.36
CNR2 P34972 3/20 0.35
CNR1 P21554 1/20 0.35
CCR5 P51681 1/20 0.35
S1PR2 O95136 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
LPAR2 Q9HBW0 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP7 Q9UHL4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7204853 0.90 LSS (0.46) HTR2ALSSPTGDR2KCNH2GPR119
SCHEMBL7204847 0.90 LSS (0.46) HTR2ALSSPTGDR2KCNH2GPR119
SCHEMBL4797970 0.80 LSS (0.58) HTR2ALSSPTGDR2
SCHEMBL4797966 0.80 LSS (0.58) HTR2ALSSPTGDR2
SCHEMBL27578416 0.77 LSS (0.44) HTR2ALSSPTGDR2KCNH2GPR119
SCHEMBL27578415 0.77 LSS (0.44) HTR2ALSSPTGDR2KCNH2GPR119
SCHEMBL7206605 0.77 LSS (0.50) HTR2ALSSPTGDR2KCNH2ALDH1A1
SCHEMBL7206600 0.77 LSS (0.50) HTR2ALSSPTGDR2KCNH2ALDH1A1
SCHEMBL7208943 0.76 LSS (0.45) HTR2ALSS
SCHEMBL7206164 0.75 MCHR1 (0.46) LSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1311475-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-05-21 EP disclosed
WO-2002014267-A1 NOVEL AMINOCYCLOHEXANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-02-21 WO disclosed