SCHEMBL7205103

SCHEMBL7205103

Nc1nc(SCc2ccccc2)nc2c1nc(Br)n2Cc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.60
ADORA1 P30542 5/20 0.60
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
TMIGD3 P0DMS9 3/20 0.46
ADORA2B P29275 3/20 0.46
CXCR2 P25025 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
HSP90AA1 P07900 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7204591 0.89 ADORA2A (0.58) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL5161492 0.89 TSHR (0.53) ADORA2AADORA1RAB9ASMN1; SMN2NPC1
SCHEMBL7205682 0.87 ADORA2A (0.56) ADORA2AADORA1TMIGD3ADORA2BMAPK1
SCHEMBL7211495 0.86 ADORA2A (0.61) ADORA2AADORA1TMIGD3ADORA2BTSHR
SCHEMBL7210266 0.86 ADORA2A (0.61) ADORA2AADORA1SMN1; SMN2TMIGD3ADORA2B
SCHEMBL7208531 0.86 ADORA2A (0.55) ADORA2AADORA1RAB9ATMIGD3ADORA2B
SCHEMBL7208339 0.85 ADORA3 (0.48) ADORA2AADORA1RAB9ASMN1; SMN2NPC1
SCHEMBL7205585 0.85 ADORA2A (0.54) ADORA2AADORA1TMIGD3ADORA2B
SCHEMBL7206709 0.84 ADORA2A (0.53) ADORA2AADORA1TMIGD3ADORA2B
SCHEMBL7205857 0.84 ADORA2A (0.53) ADORA2AADORA1TMIGD3ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1035123-B1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMA (JP) 2003-08-20 EP disclosed
US-6329381-B1 INTERFERONS, VIRICIDES AND ANTICARCINOGENIC AGENTS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2001-12-11 US disclosed
EP-1035123-A1 NOVEL HETEROCYCLIC COMPOUNDS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-09-13 EP disclosed